Iodide

Iodide

SCHEMBL2016304

Cn1c(COC(=O)c2nc(Cl)c(N)nc2N)[n+](C)c2ccc(Br)cc21.[I-]

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GABRA2 P47869 2/20 0.32
GABRB2 P47870 2/20 0.32
LMNA P02545 1/20 0.32
PDGFRA P16234 1/20 0.31
CDK5 Q00535 1/20 0.31
TYRO3 Q06418 1/20 0.31
RECQL P46063 1/20 0.30
KMT2A Q03164 1/20 0.30
ELANE P08246 1/20 0.30
SCNN1A P37088 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12635720 0.99 GABRA2 (0.32) GABRA2GABRB2LMNAPDGFRACDK5
Iodide SCHEMBL2021198 0.90 MAPT (0.36) GABRA2GABRB2LMNA
Iodide SCHEMBL2017463 0.89 KDM4E (0.33) GABRA2GABRB2LMNARECQLKMT2A
SCHEMBL12635733 0.89 MAPT (0.36) GABRA2GABRB2LMNA
Iodide SCHEMBL2014821 0.89 KDM4E (0.33) GABRA2GABRB2LMNAPDGFRACDK5
Iodide SCHEMBL2016658 0.88 SCNN1A (0.38) GABRA2GABRB2LMNAKMT2ASCNN1A
SCHEMBL12636299 0.88 ALDH1A1 (0.33) GABRA2GABRB2LMNAPDGFRACDK5
Iodide SCHEMBL2016067 0.86 TDP1 (0.34) GABRA2LMNAELANESCNN1A
Iodide SCHEMBL2016509 0.85 SCNN1A (0.39) GABRA2GABRB2LMNAKMT2ASCNN1A
SCHEMBL12635715 0.85 LMNA (0.44) GABRA2GABRB2LMNARECQLKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO claimed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed