SCHEMBL2016532

SCHEMBL2016532

NS(=O)(=O)c1ccc(CNC(=O)C2CCC(c3ccccc3)N(S(=O)(=O)c3ccccc3)C2)cc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA1 P00915 9/20 0.54
CA2 P00918 9/20 0.54
CA9 Q16790 8/20 0.54
CA12 O43570 5/20 0.54
ALDH1A1 P00352 4/20 0.53
MAPK1 P28482 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
FKBP1A P62942 1/20 0.48
KMT2A Q03164 2/20 0.47
RAB9A P51151 1/20 0.47
CA7 P43166 3/20 0.47
CA5A P35218 1/20 0.46
CA5B Q9Y2D0 1/20 0.46
MEN1 O00255 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12628953 1.00 CA1 (0.54) CA1CA2CA9CA12ALDH1A1
SCHEMBL2011504 0.92 ALDH1A1 (0.54) ALDH1A1NPSR1FKBP1AKMT2ARAB9A
SCHEMBL12628159 0.92 ALDH1A1 (0.54) ALDH1A1NPSR1FKBP1AKMT2ARAB9A
SCHEMBL2013800 0.91 ALDH1A1 (0.52) CA1CA2CA9CA12ALDH1A1
SCHEMBL12628186 0.91 ALDH1A1 (0.52) CA1CA2CA9CA12ALDH1A1
SCHEMBL2017637 0.89 ALDH1A1 (0.66) ALDH1A1KMT2ARAB9AMEN1
SCHEMBL12629084 0.89 ALDH1A1 (0.66) ALDH1A1KMT2ARAB9AMEN1
SCHEMBL2010853 0.89 KMT2A (0.58) ALDH1A1KMT2ARAB9AMEN1
SCHEMBL12628174 0.89 KMT2A (0.58) ALDH1A1KMT2ARAB9AMEN1
SCHEMBL12628167 0.87 ALDH1A1 (0.50) ALDH1A1FKBP1AKMT2ARAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073269-A1 PIPERIDINE ARYL SULFONAMIDE DERIVATIVES AS KV1.3 MODULATORS EVOTEC AG (DE) 2011-06-23 WO claimed