SCHEMBL20171110

SCHEMBL20171110

Cc1cccc2c(NC(C)O)cccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.50
CYP2A6 P11509 2/20 0.50
IDO1 P14902 2/20 0.42
ALDH1A1 P00352 4/20 0.39
CA12 O43570 1/20 0.35
CA2 P00918 1/20 0.35
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
MMP8 P22894 1/20 0.35
MMP14 P50281 1/20 0.35
CA14 Q9ULX7 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
PSMD14 O00487 1/20 0.34
COPS5 Q92905 1/20 0.34
HIF1A Q16665 1/20 0.33
EPAS1 Q99814 1/20 0.33
HPGD P15428 1/20 0.33
PARP1 P09874 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11405726 0.81 IDO1 (0.59) IDO1ALDH1A1HPGD
SCHEMBL11454361 0.80 MAPT (0.46) CYP1A2ALDH1A1NPC1RAB9AHIF1A
SCHEMBL2230553 0.79 NPC1 (0.48) ALDH1A1NPC1RAB9AHPGDHTT
SCHEMBL26385190 0.79 NPC1 (0.48) ALDH1A1NPC1RAB9AHPGDHTT
SCHEMBL4050170 0.78 ALDH1A1 (0.50) CYP1A2ALDH1A1CA2NPC1RAB9A
SCHEMBL11336488 0.78 CA12 (0.56) CYP1A2ALDH1A1CA12CA2MMP2
SCHEMBL143227 0.77 ALDH1A1 (0.34) CYP1A2IDO1ALDH1A1CA2NPC1
SCHEMBL11707890 0.74 KDM4E (0.38) CYP1A2ALDH1A1NPC1RAB9ACYP2C9
SCHEMBL19848459 0.73 SIGMAR1 (0.39) ALDH1A1NPC1RAB9AHPGDCYP2C9
SCHEMBL1004808 0.73 ALDH1A1 (0.40) CYP1A2CYP2A6ALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2772480-B2 HIV REPLICATION INHIBITOR SHIONOGI & CO (JP) 2020-12-09 EP disclosed
EP-2772480-B1 HIV REPLICATION INHIBITOR SHIONOGI & CO (JP) 2018-05-23 EP disclosed