SCHEMBL20171993

SCHEMBL20171993

Cc1ccc(-c2ccc(N)nc2C)c(C)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.52
NOS2 P35228 3/20 0.52
NOS1 P29475 2/20 0.52
BACE1 P56817 2/20 0.48
NCK1 P16333 1/20 0.48
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 4/20 0.43
MAPT P10636 3/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
HPGD P15428 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
FGFR1 P11362 1/20 0.40
FGFR2 P21802 1/20 0.40
CTSD P07339 1/20 0.39
GABRP O00591 1/20 0.39
GABRD O14764 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRG2 P18507 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19390798 0.81 ESR2 (0.55) NOS3NOS2NOS1ALDH1A1KDM4E
SCHEMBL4488580 0.81 NOS3 (0.48) NOS3NOS2NOS1BACE1NCK1
SCHEMBL17178279 0.79 NCF1 (0.51) NOS3NOS2NOS1ALDH1A1KDM4E
SCHEMBL4581787 0.76 NOS3 (0.50) NOS3NOS2NOS1BACE1NCK1
SCHEMBL31547677 0.76 TDP1 (0.52) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL3043421 0.76 TDP1 (0.52) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL11438697 0.75 DRD1 (0.39) NOS3NOS2NOS1BACE1NCK1
SCHEMBL17174290 0.75 NOS3 (0.42) NOS3NOS2NOS1BACE1KDM4E
SCHEMBL4581864 0.74 RAB9A (0.51) NOS3NOS2NOS1BACE1NCK1
SCHEMBL4496629 0.73 NOS3 (0.52) NOS3NOS2NOS1BACE1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3323821-A1 HETEROAROMATIC COMPOUNDS AND THEIR USE AS DOPAMINE D1 LIGANDS Pfizer Inc (US) 2018-05-23 EP disclosed