SCHEMBL11438697

SCHEMBL11438697

Cc1ccc(-c2ncc(N)nc2C)c(C)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 1/20 0.39
KDM4E B2RXH2 3/20 0.39
MAPT P10636 3/20 0.39
ALDH1A1 P00352 3/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HPGD P15428 1/20 0.39
HSP90AB1 P08238 2/20 0.38
NOS3 P29474 5/20 0.37
NOS2 P35228 5/20 0.37
NOS1 P29475 4/20 0.37
FGFR1 P11362 1/20 0.37
FGFR2 P21802 1/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
BACE1 P56817 2/20 0.36
NCK1 P16333 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
CRHR1 P34998 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17263289 0.83 JAK3 (0.46) KDM4EMAPTALDH1A1NPC1RAB9A
SCHEMBL11367319 0.79 ADORA2A (0.46) NOS3NOS2NOS1KMT2ABACE1
SCHEMBL11369575 0.75 SMN1; SMN2 (0.44) KDM4EMAPTALDH1A1SMN1; SMN2NOS3
SCHEMBL20171993 0.75 NOS3 (0.52) KDM4EMAPTALDH1A1NPC1RAB9A
SCHEMBL18356854 0.74 CNR2 (0.44) MAPTNPC1RAB9AHSP90AB1NOS3
SCHEMBL15803778 0.73 ADORA1 (0.50) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL17263278 0.73 HSP90AB1 (0.39) KDM4EMAPTALDH1A1NPC1RAB9A
SCHEMBL20171948 0.72 HSP90AB1 (0.37) DRD1KDM4EMAPTALDH1A1NPC1
SCHEMBL14483985 0.72 HTR5A (0.38) KDM4EMAPTALDH1A1NPC1RAB9A
SCHEMBL11376072 0.72 FEN1 (0.51) NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0018144-A1 A process for the preparation of substituted 2-aminopyrazines ELI LILLY AND COMPANY (US) 1980-10-29 EP disclosed
US-4211870-A FROM AMINOACETONITRILE AND A PHENYL A-HALO OXIME ELI LILLY AND COMPANY (US) 1980-07-08 US disclosed