SCHEMBL20172444

SCHEMBL20172444

Clc1ccc(Nc2cccnc2)nc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.54
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
RAB9A P51151 1/20 0.47
NPC1 O15118 1/20 0.47
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
ADRA2A P08913 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
NAMPT P43490 1/20 0.44
CYP19A1 P11511 1/20 0.44
PDE10A Q9Y233 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KDR P35968 1/20 0.43
EGFR P00533 1/20 0.43
TNNI3K Q59H18 1/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21258720 0.82 HCAR3 (0.56) MEN1KMT2ARAB9ANPC1L3MBTL1
SCHEMBL20172471 0.79 NPC1 (0.47) MEN1KMT2ARAB9ANPC1CYP11B1
SCHEMBL20172469 0.78 KMT2A (0.62) SMN1; SMN2MEN1KMT2ARAB9ANPC1
SCHEMBL31240789 0.78 ABL1 (0.48) MEN1KMT2ARAB9AALDH1A1LMNA
SCHEMBL4650666 0.78 GRM5 (0.77) SMN1; SMN2RAB9ANAMPTALDH1A1
SCHEMBL28402729 0.77 MAPT (0.57) ADRA2AADRA2BADRA2CL3MBTL1MAPT
SCHEMBL29501822 0.77 MAPT (0.57) ADRA2AADRA2BADRA2CL3MBTL1MAPT
SCHEMBL3951733 0.77 MEN1 (0.63) MEN1KMT2ARAB9ANPC1KDR
SCHEMBL4037525 0.77 TSHR (0.61) SMN1; SMN2MEN1KMT2ARAB9ANPC1
SCHEMBL22655182 0.76 ALDH1A1 (0.66) MEN1KMT2ARAB9ANPC1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106255688-B Morpholine-pyridine derivate 豪夫迈·罗氏有限公司 2019-11-08 CN disclosed
EP-3137459-B1 MORPHOLIN-PYRIDINE DERIVATIVES HAVING AFFINITY TO THE TAAR1 RECEPTOR HOFFMANN LA ROCHE (CH) 2018-05-23 EP disclosed