SCHEMBL20173781

SCHEMBL20173781

CNCCCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](CC(C)C)NC(=O)OC(C)(C)C)C(=O)OC

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 8/20 0.47
ITGA2B P08514 8/20 0.47
KMT2A Q03164 1/20 0.46
F2 P00734 1/20 0.44
PRSS1 P07477 1/20 0.44
HDAC1 Q13547 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
MAPK1 P28482 1/20 0.41
CMA1 P23946 6/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20174121 0.89 F2 (0.54) F2PRSS1MAPK1CMA1
SCHEMBL20173779 0.84 KMT2A (0.48) ITGB3ITGA2BKMT2AF2PRSS1
SCHEMBL11661759 0.79 KMT2A (0.64) KMT2AALDH1A1LMNA
SCHEMBL31186061 0.79 KMT2A (0.64) KMT2AALDH1A1LMNA
SCHEMBL3046422 0.79 KMT2A (0.64) KMT2AALDH1A1LMNA
SCHEMBL20174122 0.79 OPRK1 (0.61) F2
SCHEMBL23832913 0.78 ACE (0.55) KMT2AF2MAPK1CMA1ALDH1A1
SCHEMBL2262043 0.78 ACE (0.55) KMT2AF2MAPK1CMA1ALDH1A1
SCHEMBL10935144 0.78 ACE (0.55) KMT2AF2MAPK1CMA1ALDH1A1
SCHEMBL9510956 0.77 KMT2A (0.52) KMT2AF2PRSS1HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094335-A1 FINE-TUNE MODULATORS OF NEURONAL EXCITABILITY FOR NEUROPSYCHIATRIC DISORDERS THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2018-05-24 WO disclosed