SCHEMBL20176626

SCHEMBL20176626

NC(=O)c1cncc(Oc2ccc(Br)cc2)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 7/20 0.65
SIRT3 Q9NTG7 7/20 0.65
SIRT1 Q96EB6 6/20 0.65
PARP10 Q53GL7 8/20 0.50
PARP15 Q460N3 4/20 0.50
PARP14 Q460N5 2/20 0.50
ALDH1A1 P00352 1/20 0.50
KMT2A Q03164 1/20 0.50
PARP16 Q8N5Y8 1/20 0.50
PARP11 Q9NR21 1/20 0.50
PARP4 Q9UKK3 1/20 0.50
CDC7 O00311 1/20 0.50
DYRK3 O43781 1/20 0.50
ROCK2 O75116 1/20 0.50
MAP4K4 O95819 1/20 0.50
ICAM1 P05362 1/20 0.50
FYN P06241 1/20 0.50
CDK1 P06493 1/20 0.50
PIM1 P11309 1/20 0.50
SELE P16581 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28281436 0.86 SIRT2 (0.76) SIRT2SIRT3SIRT1PARP10PARP15
SCHEMBL9926362 0.84 SIRT2 (0.65) SIRT2SIRT3SIRT1PARP10PARP15
SCHEMBL20176625 0.82 ATM (0.51) SIRT2SIRT3SIRT1ALDH1A1KMT2A
SCHEMBL15314416 0.79 SIRT2 (0.57) SIRT2SIRT3SIRT1PARP10PARP15
SCHEMBL3698084 0.76 SIRT2 (0.54) SIRT2SIRT3SIRT1ROCK1
SCHEMBL31137907 0.74 POLB (0.67) SIRT2SIRT3SIRT1ALDH1A1KMT2A
SCHEMBL578591 0.74 POLB (0.67) SIRT2SIRT3SIRT1ALDH1A1KMT2A
SCHEMBL28068268 0.73 PARP15 (0.55) SIRT2SIRT3SIRT1PARP10PARP15
SCHEMBL9448469 0.73 MKNK1 (0.66) SIRT2SIRT3SIRT1PARP10PARP4
SCHEMBL28347899 0.73 SIRT2 (0.54) SIRT2SIRT3SIRT1KMT2AMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092047-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE JOINT STOCK COMPANY "BIOCAD" (RU) 2018-05-24 WO disclosed