SCHEMBL20177902

SCHEMBL20177902

Nc1ccccc1N1C[C@@H](c2c(F)cc(Br)cc2F)CC1=O

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.39
GRM5 P41594 1/20 0.39
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
BPTF Q12830 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177834 0.84 PDE4A (0.44) GRM4GRM5PDE4APDE4BPDE4C
SCHEMBL20177851 0.79 BRD4 (0.54) PDE4APDE4BPDE4CPDE4D
SCHEMBL20177560 0.68 ALDH1A1 (0.43) GRM5PDE4APDE4BPDE4CPDE4D
SCHEMBL20177564 0.61 KDM1A (0.32)
SCHEMBL20177500 0.61 DPP4 (0.43)
SCHEMBL17514687 0.61 KDM1A (0.35) KMT2A
SCHEMBL20177653 0.61 GSK3B (0.48) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL18640812 0.60 BPTF (0.44) GRM5PDE4APDE4BPDE4CPDE4D
SCHEMBL20177816 0.59 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL20177572 0.59 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed