SCHEMBL20177640

SCHEMBL20177640

N[C@@H]1c2nc3ccccc3n2C[C@H]1c1c(F)cc(Br)cc1F

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.38
DPP7 Q9UHL4 1/20 0.38
USP2 O75604 1/20 0.38
KDM4E B2RXH2 2/20 0.36
KDM1A O60341 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HTT P42858 1/20 0.35
RECQL P46063 1/20 0.34
PDE10A Q9Y233 1/20 0.33
TP53 P04637 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177583 0.85 FPR1 (0.41) DPP4DPP7USP2KDM4EMEN1
SCHEMBL20177495 0.80 USP2 (0.40) USP2KDM4EKDM1AMEN1KMT2A
SCHEMBL20177563 0.74 FPR2 (0.45) HTTTP53ALDH1A1
SCHEMBL20177500 0.72 DPP4 (0.43) DPP4DPP7KDM4ETP53TSHR
SCHEMBL20177499 0.69 SMN1; SMN2 (0.37) KDM4EHTTALDH1A1
SCHEMBL20177936 0.68 KDM1A (0.32) KDM1A
SCHEMBL20177716 0.68 KDM1A (0.34) KDM1A
SCHEMBL20177616 0.62 FPR2 (0.42) KDM1A
SCHEMBL13342393 0.61 DPP4 (0.82) DPP4DPP7
SCHEMBL28581918 0.61 USP2 (0.51) USP2KDM4EMEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed