SCHEMBL20177552

SCHEMBL20177552

COc1ccc(COC(=O)N[C@@H]2C(=S)NC[C@H]2c2ccc3c(c2)CCO3)cc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 1/20 0.40
NAAA Q02083 3/20 0.38
PKM P14618 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
MTNR1A P48039 2/20 0.37
ASAH1 Q13510 1/20 0.36
RYR2 Q92736 1/20 0.36
TP53 P04637 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KCNQ2 O43526 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177810 0.91 FPR1 (0.44) EDNRBNAAAASAH1
SCHEMBL20177800 0.84 EDNRB (0.38) EDNRBNAAAPKMHTTSMN1; SMN2
SCHEMBL20177571 0.81 EDNRB (0.38) EDNRBNAAAPKMHTTSMN1; SMN2
SCHEMBL20177637 0.81 FPR1 (0.44) NAAAPKMHTTSMN1; SMN2KMT2A
SCHEMBL20177949 0.81 FPR1 (0.52) NAAAPKMHTTSMN1; SMN2ASAH1
SCHEMBL20177489 0.78 FPR2 (0.44) EDNRBPKMHTTSMN1; SMN2MEN1
SCHEMBL20177658 0.76 FPR2 (0.48) NAAAPKMHTTSMN1; SMN2ASAH1
SCHEMBL20177501 0.74 FPR2 (0.47) NAAAPKMHTTSMN1; SMN2ASAH1
SCHEMBL20177604 0.74 FPR2 (0.47) NAAAPKMHTTSMN1; SMN2ASAH1
SCHEMBL20177669 0.73 FPR1 (0.43) NAAAPKMHTTSMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed