SCHEMBL20177577

SCHEMBL20177577

OCCO/N=C1/C[C@H](c2ccc(Cl)cc2F)CN1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 1/20 0.36
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
OPRL1 P41146 6/20 0.34
FPR1 P21462 1/20 0.32
FPR2 P25090 1/20 0.32
TRPM5 Q9NZQ8 3/20 0.32
TRPM4 Q8TD43 2/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNA4 P43681 1/20 0.31
PROKR1 Q8TCW9 1/20 0.31
GRM5 P41594 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177882 0.86 KDM1A (0.35)
SCHEMBL20177736 0.85 KDM1A (0.34) TRPM5
SCHEMBL20177903 0.84
SCHEMBL20177509 0.84 GPBAR1 (0.34) GPBAR1HTR2AHTR2CHTR2BOPRL1
SCHEMBL20177943 0.80 HTR3A (0.36) GPBAR1GRM5
SCHEMBL20177686 0.77
SCHEMBL19559541 0.75 FPR2 (0.34) FPR2
SCHEMBL20177855 0.75
SCHEMBL16785344 0.73 FPR1 (0.35) FPR1FPR2
SCHEMBL18117741 0.73 FPR1 (0.35) FPR1FPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed