SCHEMBL20177600

SCHEMBL20177600

O=C1C[C@H](c2ccc(Br)cc2F)CN1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.48
KDM1A O60341 2/20 0.45
KDM1B Q8NB78 1/20 0.45
PDE4A P27815 6/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
TSHR P16473 1/20 0.39
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
FPR1 P21462 1/20 0.35
FPR2 P25090 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15549178 0.84 MTNR1A (0.50) MTNR1APDE4APDE4BPDE4CPDE4D
SCHEMBL20177675 0.81 KDM1A (0.45) KDM1AKDM1BMEN1LMNAKMT2A
SCHEMBL20177704 0.81 MTNR1A (0.48) MTNR1APDE4APDE4BPDE4CPDE4D
SCHEMBL18590494 0.81 MTNR1A (0.48) MTNR1APDE4APDE4BPDE4CPDE4D
SCHEMBL20177816 0.79 PDE4A (0.39) MTNR1APDE4APDE4BPDE4CPDE4D
SCHEMBL20177572 0.79 PDE4A (0.39) MTNR1APDE4APDE4BPDE4CPDE4D
SCHEMBL30021045 0.78 KDM1A (0.56) KDM1AKDM1BCYP1A2MEN1LMNA
SCHEMBL29869025 0.78 MTNR1A (0.46) MTNR1APDE4APDE4BPDE4CPDE4D
SCHEMBL22778088 0.78 KDM1A (0.56) KDM1AKDM1BCYP1A2MEN1LMNA
SCHEMBL19559399 0.78 MTNR1A (0.64) MTNR1APDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed