SCHEMBL20179243

SCHEMBL20179243

CC(=O)Oc1ccc(CONC(=O)CCC(Cc2ccc(C(=O)OC(C)(C)C)cc2)C(=O)OC(C)(C)C)cc1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 4/20 0.42
LTA4H P09960 1/20 0.39
CACNA1B Q00975 6/20 0.36
SLC7A5 Q01650 1/20 0.35
ELANE P08246 2/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20168306 0.94 FOLH1 (0.42) FOLH1LTA4HCACNA1BLMNAPOLB
SCHEMBL20168291 0.92 FOLH1 (0.50) FOLH1LTA4HCACNA1BELANELMNA
SCHEMBL20179186 0.90 SLC7A5 (0.49) FOLH1LTA4HCACNA1BSLC7A5LMNA
SCHEMBL21577924 0.89 PRSS1 (0.38) FOLH1LTA4HCACNA1BSLC7A5ELANE
SCHEMBL20179173 0.87 SLC7A5 (0.44) FOLH1LTA4HCACNA1BSLC7A5LMNA
SCHEMBL20179151 0.85 FOLH1 (0.44) FOLH1LMNANPC1
SCHEMBL20179259 0.85 FOLH1 (0.39) FOLH1LTA4HCACNA1BSLC7A5ELANE
SCHEMBL20168691 0.84 FOLH1 (0.47) FOLH1LTA4HSLC7A5LMNARAB9A
SCHEMBL23710339 0.84 FOLH1 (0.45) FOLH1LTA4HSLC7A5LMNANPC1
SCHEMBL20179205 0.83 FOLH1 (0.52) FOLH1LMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11866394-B2 Prodrugs of hydroxamate-based GCPII inhibitors THE JOHNS HOPKINS UNIVERSTY (US) 2024-01-09 US disclosed
US-20210355079-A1 PRODRUGS OF HYDROXAMATE-BASED GCPII INHIBITORS INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY AS CR V.V.I. (CZ) 2021-11-18 US disclosed
US-11059775-B2 Prodrug compositions and utility of hydroxamate-based GCPII inhibitors THE JOHNS HOPKINS UNIVERSITY (US) 2021-07-13 US disclosed
US-20190352255-A1 NOVEL PRODRUG COMPOSITIONS AND UTILITY OF HYDROXAMATE-BASED GCPII INHIBITORS THE JOHNS HOPKINS UNIVERSITY 2019-11-21 US disclosed
WO-2018094334-A1 PRODRUGS OF HYDROXAMATE-BASED GCPII INHIBITORS THE JOHNS HOPKINS UNIVERSITY (US) 2018-05-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190352255-A1 NOVEL PRODRUG COMPOSITIONS AND UTILITY OF HYDROXAMATE-BASED GCPII INHIBITORS GPI, TPI1, HPGDS FOLH1 10/4885LTA4H 1303/4885CACNA1B 4072/4885
US-20210355079-A1 PRODRUGS OF HYDROXAMATE-BASED GCPII INHIBITORS TPI1, HPGDS, GPI FOLH1 39/4885LTA4H 1571/4885CACNA1B 4030/4885
US-11059775-B2 Prodrug compositions and utility of hydroxamate-based GCPII inhibitors GLS, HPGDS, GPI FOLH1 15/4885LTA4H 1594/4885CACNA1B 3913/4885
US-11866394-B2 Prodrugs of hydroxamate-based GCPII inhibitors TPI1, HPGDS, GPI FOLH1 39/4885LTA4H 1571/4885CACNA1B 4030/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.