SCHEMBL20168291

SCHEMBL20168291

CC(=O)Oc1ccc(CONC(=O)CCC(Cc2ccc(C(=O)O)cc2)C(=O)OC(C)(C)C)cc1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 5/20 0.50
LTA4H P09960 1/20 0.41
HSD17B10 Q99714 1/20 0.40
RXRA P19793 3/20 0.38
RXRB P28702 3/20 0.38
NR4A2 P43354 1/20 0.38
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
POLB P06746 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CACNA1B Q00975 1/20 0.34
ELANE P08246 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20179243 0.92 FOLH1 (0.42) FOLH1LTA4HNPC1RAB9APOLB
SCHEMBL20168691 0.90 FOLH1 (0.47) FOLH1LTA4HNR4A2RAB9ASMN1; SMN2
SCHEMBL20168306 0.90 FOLH1 (0.42) FOLH1LTA4HNPC1POLBSMN1; SMN2
SCHEMBL20168729 0.89 FOLH1 (0.62) FOLH1HSD17B10RXRARXRBNPC1
SCHEMBL21570571 0.87 LMNA (0.46) FOLH1LTA4HRXRANR4A2LMNA
SCHEMBL20168587 0.85 FOLH1 (0.50) FOLH1LTA4H
SCHEMBL20179186 0.84 SLC7A5 (0.49) FOLH1LTA4HRAB9ACACNA1BLMNA
SCHEMBL21577913 0.84 FOLH1 (0.48) FOLH1HSD17B10RXRARXRBNPC1
SCHEMBL20179173 0.82 SLC7A5 (0.44) FOLH1LTA4HRXRACACNA1BLMNA
SCHEMBL21577924 0.82 PRSS1 (0.38) FOLH1LTA4HNPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11866394-B2 Prodrugs of hydroxamate-based GCPII inhibitors THE JOHNS HOPKINS UNIVERSTY (US) 2024-01-09 US disclosed
US-20210355079-A1 PRODRUGS OF HYDROXAMATE-BASED GCPII INHIBITORS INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY AS CR V.V.I. (CZ) 2021-11-18 US disclosed
US-11059775-B2 Prodrug compositions and utility of hydroxamate-based GCPII inhibitors THE JOHNS HOPKINS UNIVERSITY (US) 2021-07-13 US disclosed
US-20190352255-A1 NOVEL PRODRUG COMPOSITIONS AND UTILITY OF HYDROXAMATE-BASED GCPII INHIBITORS THE JOHNS HOPKINS UNIVERSITY 2019-11-21 US disclosed
WO-2018094334-A1 PRODRUGS OF HYDROXAMATE-BASED GCPII INHIBITORS THE JOHNS HOPKINS UNIVERSITY (US) 2018-05-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190352255-A1 NOVEL PRODRUG COMPOSITIONS AND UTILITY OF HYDROXAMATE-BASED GCPII INHIBITORS GPI, TPI1, HPGDS FOLH1 10/4885LTA4H 1303/4885HSD17B10 344/4885
US-20210355079-A1 PRODRUGS OF HYDROXAMATE-BASED GCPII INHIBITORS TPI1, HPGDS, GPI FOLH1 39/4885LTA4H 1571/4885HSD17B10 361/4885
US-11059775-B2 Prodrug compositions and utility of hydroxamate-based GCPII inhibitors GLS, HPGDS, GPI FOLH1 15/4885LTA4H 1594/4885HSD17B10 403/4885
US-11866394-B2 Prodrugs of hydroxamate-based GCPII inhibitors TPI1, HPGDS, GPI FOLH1 39/4885LTA4H 1571/4885HSD17B10 361/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.