SCHEMBL20179256

SCHEMBL20179256

Cc1oc(=O)oc1CONC(=O)CCC(Cc1ccc(C(O)O)cc1)C(=O)O

nearest known ligand 0.80

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 5/20 0.80
CPA3 P15088 1/20 0.35
KDM4E B2RXH2 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CHRM1 P11229 1/20 0.31
TBXA2R P21731 1/20 0.31
ADRA1A P35348 1/20 0.31
PTGES O14684 1/20 0.31
ALOX5 P09917 1/20 0.31
PPARG P37231 1/20 0.31
PPARA Q07869 1/20 0.31
PRSS1 P07477 1/20 0.31
TMPRSS15 P98073 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24023410 0.90 FOLH1 (0.74) FOLH1CPA3KDM4ETSHRHSD17B10
SCHEMBL20179147 0.89 FOLH1 (1.00) FOLH1CPA3PPARGPRSS1TMPRSS15
SCHEMBL20179133 0.86 FOLH1 (0.82) FOLH1KDM4ETSHRHSD17B10PPARG
SCHEMBL21578051 0.85 FOLH1 (0.75) FOLH1CPA3KDM4ETSHRHSD17B10
SCHEMBL26039286 0.82 FOLH1 (0.63) FOLH1PPARG
SCHEMBL20179142 0.79 FOLH1 (0.72) FOLH1TSHRPPARGPPARA
SCHEMBL21570573 0.79 FOLH1 (0.80) FOLH1
SCHEMBL21577914 0.78 FOLH1 (0.80) FOLH1PRSS1TMPRSS15
SCHEMBL26038808 0.76 FOLH1 (0.76) FOLH1
SCHEMBL20168739 0.75 FOLH1 (0.66) FOLH1KDM4ETSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11059775-B2 Prodrug compositions and utility of hydroxamate-based GCPII inhibitors THE JOHNS HOPKINS UNIVERSITY (US) 2021-07-13 US disclosed
US-20190352255-A1 NOVEL PRODRUG COMPOSITIONS AND UTILITY OF HYDROXAMATE-BASED GCPII INHIBITORS THE JOHNS HOPKINS UNIVERSITY 2019-11-21 US disclosed
WO-2018094334-A1 PRODRUGS OF HYDROXAMATE-BASED GCPII INHIBITORS THE JOHNS HOPKINS UNIVERSITY (US) 2018-05-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190352255-A1 NOVEL PRODRUG COMPOSITIONS AND UTILITY OF HYDROXAMATE-BASED GCPII INHIBITORS GPI, TPI1, HPGDS FOLH1 10/4885CPA3 345/4885KDM4E 3355/4885
US-11059775-B2 Prodrug compositions and utility of hydroxamate-based GCPII inhibitors GLS, HPGDS, GPI FOLH1 15/4885CPA3 382/4885KDM4E 3638/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.