SCHEMBL20180369

SCHEMBL20180369

O=Cc1ccc2c(-c3ccccc3Cl)cn(-c3ccc(F)cc3)c2c1

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DGAT2 Q96PD7 16/20 0.52
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 1/20 0.44
RORC P51449 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28309854 0.81 ALDH1A1 (0.52) DGAT2ALDH1A1KDM4ERORC
SCHEMBL20180267 0.77 DGAT2 (0.51) DGAT2ALDH1A1RORC
SCHEMBL20166496 0.77 DGAT2 (0.70) DGAT2
SCHEMBL20180470 0.69 DGAT2 (1.00) DGAT2
SCHEMBL20180282 0.69 DGAT2 (0.73) DGAT2
SCHEMBL5896326 0.69 ALDH1A1 (0.46) ALDH1A1
SCHEMBL26122642 0.68 ALDH1A1 (0.57) ALDH1A1KDM4E
SCHEMBL31632773 0.67 SCN9A (0.44) ALDH1A1KDM4E
SCHEMBL3716522 0.67 ALDH1A1 (1.00) ALDH1A1KDM4E
SCHEMBL12810492 0.66 HTR6 (0.52) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018093698-A1 INDOLE DERIVATIVES USEFUL AS INHIBITORS OF DIACYLGLYCERIDE O-ACYLTRANSFERASE 2 MERCK SHARP & DOHME CORP. (US) 2018-05-24 WO disclosed