SCHEMBL20180640

SCHEMBL20180640

Cc1c(-c2cccc(OC(F)F)c2)c2ccc(C=O)cc2n1-c1ccc(F)cc1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DGAT2 Q96PD7 8/20 0.57
DRD1 P21728 3/20 0.49
PPARG P37231 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
TP53 P04637 1/20 0.33
THRB P10828 1/20 0.33
HTT P42858 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20180267 0.76 DGAT2 (0.51) DGAT2TP53
SCHEMBL20166221 0.73 DGAT2 (1.00) DGAT2
SCHEMBL12334437 0.67 POLB (0.49) PPARGMAPTKDM4ETP53HTT
SCHEMBL13051741 0.66 HTT (0.46) PPARGMAPTKDM4EHTT
SCHEMBL856123 0.66 DRD1 (0.68) DRD1MAOAMAOBMAPT
SCHEMBL29391855 0.66 DRD1 (0.68) DRD1MAOAMAOBMAPT
SCHEMBL13299344 0.63 IP6K1 (0.43) KDM4E
SCHEMBL11986618 0.63 NR3C1 (0.40) DGAT2KDM4E
SCHEMBL20526641 0.62 JAK2 (0.48) KDM4EHTT
SCHEMBL12489894 0.62 POLB (0.51) PPARGMAPTKDM4ETP53HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018093698-A1 INDOLE DERIVATIVES USEFUL AS INHIBITORS OF DIACYLGLYCERIDE O-ACYLTRANSFERASE 2 MERCK SHARP & DOHME CORP. (US) 2018-05-24 WO disclosed