SCHEMBL20181869

SCHEMBL20181869

Cc1cn(Cc2cnc(-c3ccccc3F)[nH]2)c2ncnc(Cl)c12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NR2F2 P24468 1/20 0.36
ACP1 P24666 2/20 0.35
MAPK13 O15264 4/20 0.34
MAPK12 P53778 4/20 0.34
MAPK11 Q15759 4/20 0.34
MAPK14 Q16539 4/20 0.34
CXCR2 P25025 1/20 0.33
MGAM O43451 1/20 0.33
GAA P10253 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
SRC P12931 1/20 0.32
GRIN2B Q13224 4/20 0.32
ADK P55263 1/20 0.31
KCNH2 Q12809 1/20 0.31
SCN5A Q14524 1/20 0.31
SCN9A Q15858 1/20 0.31
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20162739 0.88 CXCR2 (0.35) MEN1KMT2ANR2F2ACP1MAPK13
SCHEMBL30037624 0.88 CXCR2 (0.35) MEN1KMT2ANR2F2ACP1MAPK13
SCHEMBL30038073 0.78 SRC (0.47) SRC
SCHEMBL20162580 0.78 SRC (0.47) SRC
SCHEMBL20162902 0.78 DYRK3 (0.41) SRC
SCHEMBL30037066 0.78 DYRK3 (0.41) SRC
SCHEMBL20181875 0.77 RET (0.34) MEN1KMT2ANR2F2MAPK13MAPK12
SCHEMBL20182174 0.73 DRD2 (0.40) MEN1KMT2ANR2F2GRIN2BADK
SCHEMBL20182201 0.71 NOTUM (0.48) GRIN2BKCNH2
SCHEMBL20162748 0.70 SRC (0.43) SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed