SCHEMBL20184540

SCHEMBL20184540

O=C(O)c1c[nH]c2ncnc(-c3ccccc3Cl)c12

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 7/20 0.51
JAK3 P52333 7/20 0.51
BTK Q06187 10/20 0.46
LRRK2 Q5S007 1/20 0.44
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20184579 0.85 JAK2 (0.52) JAK2JAK3LRRK2KDM4EMEN1
SCHEMBL20184436 0.84 JAK3 (0.57) JAK2JAK3BTK
SCHEMBL20184461 0.84 JAK3 (0.69) JAK2JAK3BTKLRRK2KDM4E
SCHEMBL15032693 0.82 JAK3 (0.77) JAK2JAK3
SCHEMBL20184432 0.82 JAK3 (0.68) JAK2JAK3
SCHEMBL20184454 0.80 JAK3 (0.70) JAK2JAK3
SCHEMBL20184363 0.78 JAK3 (0.55) JAK2JAK3
SCHEMBL20184385 0.77 JAK3 (0.71) JAK2JAK3LRRK2
SCHEMBL20184403 0.77 DHODH (0.42) JAK2JAK3HSP90AB1HPGDKMT2A
SCHEMBL20184596 0.76 JAK3 (0.71) JAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2788000-B1 PYRROLOPYRIMIDINES AS JANUS KINASE INHIBITORS MERCK SHARP & DOHME (US) 2018-05-30 EP claimed