SCHEMBL20195396

SCHEMBL20195396

COc1cccc(OCc2c(Cl)cccc2N(N)C(=O)N(C)N)n1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.38
NR1H4 Q96RI1 7/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
JAK3 P52333 1/20 0.34
NFE2L2 Q16236 1/20 0.34
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22038784 0.90 HTR7 (0.41) SMN1; SMN2NR1H4NPSR1
SCHEMBL20844967 0.82 NR1H4 (0.35) SMN1; SMN2NR1H4MAPTMAPK1
SCHEMBL22038791 0.81 HTR7 (0.41) MAPTMAPK1
SCHEMBL20195405 0.78 NPSR1 (0.34) NPSR1
SCHEMBL22037708 0.78 HTR7 (0.42) NR1H4MAPT
SCHEMBL22037218 0.77 CYP3A4 (0.35) SMN1; SMN2NR1H4MAPK1
SCHEMBL22037209 0.77 NR1H4 (0.32) NR1H4RXRARXRBRXRG
SCHEMBL22037272 0.77 HTR7 (0.41)
SCHEMBL18831732 0.77 HTT (0.39) SMN1; SMN2MAPTMAPK1
SCHEMBL18831547 0.76 MAOA (0.37) SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3029035-B1 TETRAZOLINONE COMPOUND, AND USE THEREOF SUMITOMO CHEMICAL CO (JP) 2018-05-30 EP disclosed