SCHEMBL20197285

SCHEMBL20197285

CCCc1nc2c(I)ccnc2[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 8/20 0.42
GSK3B P49841 8/20 0.42
CDK1 P06493 7/20 0.42
CCNB2 O95067 6/20 0.42
CCNB1 P14635 6/20 0.42
CCNB3 Q8WWL7 6/20 0.42
CDK5 Q00535 5/20 0.42
CDK5R1 Q15078 4/20 0.42
KDM4C Q9H3R0 1/20 0.41
CDK2 P24941 3/20 0.38
MAPK8 P45983 3/20 0.38
CCNE1 P24864 2/20 0.38
CCNE2 O96020 1/20 0.38
INSR P06213 1/20 0.38
CFTR P13569 1/20 0.38
CCNA2 P20248 1/20 0.38
MAPK3 P27361 1/20 0.38
MAPK1 P28482 1/20 0.38
MAPK9 P45984 1/20 0.38
MAPK10 P53779 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1056828 0.88 ADORA3 (0.41) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL4370037 0.85 NOS2 (0.41) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL8972110 0.83 KDM4C (0.39) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL16544507 0.81 KDM4C (0.38) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1080357 0.77 CCNB2 (0.40) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL3964555 0.77 ADORA1 (0.43) KDM4CPDE3BPDE3AADORA3ADORA2A
SCHEMBL8875881 0.76 GSK3B (0.44) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL6641610 0.74 CCNB2 (0.36) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL4295424 0.74 NOS2 (0.58) GSK3AGSK3BCDK1CCNB2CCNB1
SCHEMBL1058944 0.74 CCNB2 (0.38) GSK3AGSK3BCDK1CCNB2CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3038622-B1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECH LLC (US) 2018-05-30 EP disclosed