SCHEMBL3964555

SCHEMBL3964555

CCCc1nc2nccc(I)c2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.43
ADORA3 P0DMS8 2/20 0.43
ADORA2A P29274 2/20 0.43
PI4KA P42356 1/20 0.42
PI4K2B Q8TCG2 1/20 0.42
PI4K2A Q9BTU6 1/20 0.42
PI4KB Q9UBF8 1/20 0.42
NOS2 P35228 8/20 0.42
NOS1 P29475 7/20 0.42
NOS3 P29474 4/20 0.42
KDM4C Q9H3R0 1/20 0.36
POLB P06746 1/20 0.35
CYP2C9 P11712 1/20 0.34
TACR2 P21452 1/20 0.33
KDM4E B2RXH2 1/20 0.32
KDM5A P29375 1/20 0.32
KDM5B Q9UGL1 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
HCAR2 Q8TDS4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7378689 0.82 NOS2 (0.59) ADORA1ADORA3ADORA2API4KAPI4K2B
SCHEMBL9406926 0.81 ADORA1 (0.43) ADORA1ADORA3ADORA2API4KAPI4K2B
SCHEMBL9406899 0.78 ADORA1 (0.42) ADORA1ADORA3ADORA2API4KAPI4K2B
SCHEMBL20197285 0.77 GSK3A (0.42) ADORA1ADORA3ADORA2API4KAPI4K2B
SCHEMBL3650837 0.75 KDM4E (0.45) ADORA1ADORA3ADORA2API4KAPI4K2B
SCHEMBL8561715 0.74 ADORA1 (0.41) ADORA1ADORA3ADORA2API4KAPI4K2B
SCHEMBL9041424 0.73 NOS1 (0.56) ADORA1PI4KAPI4K2BPI4K2API4KB
SCHEMBL9648738 0.72 PI4KA (0.57) ADORA1PI4KAPI4K2BPI4K2API4KB
SCHEMBL9406720 0.71 PI4KA (0.56) PI4KAPI4K2BPI4K2API4KBNOS2
SCHEMBL4052252 0.70 KDM4C (0.41) ADORA1ADORA3ADORA2API4KAPI4K2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009034411-A1 PERHARIDINES AS CDK INHIBITORS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2009-03-19 WO disclosed