SCHEMBL20201699

SCHEMBL20201699

Cc1cc(OCC2CC2)c(C)cc1F

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.40
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
HTR2B P41595 2/20 0.38
RIPK1 Q13546 1/20 0.38
RET P07949 2/20 0.38
SCN9A Q15858 3/20 0.36
BRD4 O60885 1/20 0.36
ELANE P08246 1/20 0.36
KCNN4 O15554 1/20 0.35
HPGD P15428 1/20 0.35
PDE2A O00408 1/20 0.35
CNR2 P34972 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20376455 0.89 HTR2A (0.38) PDE10AHTR2AHTR2CHTR2BRIPK1
SCHEMBL20201733 0.85 SCN9A (0.46) SCN9A
SCHEMBL21325507 0.82 HTR2C (0.40) PDE10AHTR2AHTR2CHTR2BRIPK1
SCHEMBL21325098 0.82 DHFR (0.41) PDE10AHTR2AHTR2CHTR2BRIPK1
SCHEMBL24777832 0.81 SCN9A (0.49) SCN9A
SCHEMBL9896972 0.81 SCN9A (0.36) PDE10AHTR2AHTR2CHTR2BRIPK1
SCHEMBL13475569 0.79 HPGD (0.49) ELANEHPGD
SCHEMBL18374001 0.79 HTR2C (0.51) PDE10AHTR2AHTR2CHTR2BRIPK1
SCHEMBL16135136 0.79 CYP3A4 (0.40) PDE10AHTR2AHTR2CHTR2BRIPK1
SCHEMBL20201700 0.79 ALDH1A1 (0.42) HTR2CHTR2BRIPK1RETCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018128720-A1 URACIL CONTAINING COMPOUNDS CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-07-12 WO disclosed
WO-2018098206-A1 HYDANTOIN CONTAINING DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-05-31 WO disclosed
WO-2018098208-A1 NITROGEN RING LINKED DEOXYURIDINE TRIPHOSPHATASE INHIBITORS CV6 THERAPEUTICS (NI) LIMITED (GB) 2018-05-31 WO disclosed