SCHEMBL20207639

SCHEMBL20207639

C/N=C(/Nc1c(OC)cccc1OC)c1nccs1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.41
RAB9A P51151 6/20 0.39
NPC1 O15118 5/20 0.39
ADRB2 P07550 1/20 0.39
GRM4 Q14833 1/20 0.38
KMT2A Q03164 4/20 0.37
MEN1 O00255 2/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
MAPK1 P28482 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
SNCA P37840 1/20 0.36
CTSA P10619 1/20 0.36
RBBP9 O75884 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PKM P14618 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20207359 0.88 GAA (0.41) GAARAB9ANPC1ADRB2GRM4
SCHEMBL20189542 0.88 GAA (0.41) GAARAB9ANPC1ADRB2GRM4
SCHEMBL20189540 0.88 GAA (0.41) GAARAB9ANPC1ADRB2GRM4
SCHEMBL20188746 0.81 GRM4 (0.52) GAARAB9ANPC1ADRB2GRM4
SCHEMBL20190237 0.81 GAA (0.43) GAARAB9ANPC1ADRB2GRM4
SCHEMBL20207357 0.81 GAA (0.43) GAARAB9ANPC1ADRB2GRM4
SCHEMBL15111138 0.69 SMN1; SMN2 (0.47) GAARAB9ANPC1GRM4KMT2A
SCHEMBL20180716 0.68 SMN1; SMN2 (0.49) GAARAB9ANPC1KMT2AMEN1
SCHEMBL723820 0.66 RORC (0.53) GAARAB9ANPC1ADRB2GRM4
SCHEMBL20775422 0.65 NLRP3 (0.61) GAARAB9ANPC1ADRB2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018097945-A1 HETEROARYL-SUBSTITUTED TRIAZOLES AS APJ RECEPTOR AGONISTS AMGEN INC. (US) 2018-05-31 WO disclosed