SCHEMBL20208640

SCHEMBL20208640

Cc1c(N=O)ccc2c3c(c(=O)oc12)CN(C(=O)OCc1ccccc1)CC3

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 9/20 0.49
MTHFD1 P11586 1/20 0.45
MTHFD2 P13995 1/20 0.45
TMEM97 Q5BJF2 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
PTGDR2 Q9Y5Y4 8/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21354099 0.88 ERN1 (0.58) ERN1MTHFD1MTHFD2TMEM97SIGMAR1
SCHEMBL21417110 0.82 TMEM97 (0.49) ERN1MTHFD1MTHFD2TMEM97SIGMAR1
SCHEMBL20208889 0.82 MTHFD1 (0.47) ERN1MTHFD1MTHFD2DRD2DRD4
SCHEMBL21354138 0.81 MTHFD1 (0.47) ERN1MTHFD1MTHFD2DRD2DRD4
SCHEMBL24691517 0.81 MTHFD1 (0.46) ERN1MTHFD1MTHFD2DRD2DRD4
SCHEMBL20208684 0.76 CXCR3 (0.47) ERN1MTHFD1MTHFD2TMEM97SIGMAR1
SCHEMBL23949707 0.73 TMEM97 (0.57) TMEM97SIGMAR1PTGDR2
SCHEMBL31454878 0.72 ERN1 (0.79) ERN1MTHFD1MTHFD2DRD4
SCHEMBL16197809 0.71 ERN1 (0.71) ERN1MTHFD1MTHFD2DRD2DRD4
SCHEMBL20208638 0.70 GAA (0.51) ERN1DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018097162-A1 SULFONAMIDE DERIVATIVE HAVING COUMARIN SKELETON 第一三共株式会社 2018-05-31 WO disclosed