SCHEMBL20208638

SCHEMBL20208638

Cc1c(O)ccc2c3c(c(=O)oc12)CN(C(O)OCc1ccccc1)CC3

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.51
KDM4E B2RXH2 2/20 0.51
ALDH1A1 P00352 2/20 0.51
GLA P06280 2/20 0.51
HPGD P15428 2/20 0.51
CASP1 P29466 2/20 0.51
CASP7 P55210 2/20 0.51
HSD17B10 Q99714 2/20 0.51
MAOA P21397 1/20 0.51
MAPK1 P28482 1/20 0.51
ERN1 O75460 6/20 0.50
SHBG P04278 1/20 0.47
DRD4 P21917 4/20 0.46
DRD2 P14416 3/20 0.46
DRD3 P35462 3/20 0.46
LMNA P02545 1/20 0.43
ESR2 Q92731 1/20 0.43
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20208888 0.83 DRD2 (0.44) KDM4EALDH1A1HPGDHSD17B10MAOA
SCHEMBL20208640 0.70 ERN1 (0.49) ERN1DRD4DRD2DRD3
SCHEMBL20208562 0.69 KDM4E (0.55) GAAKDM4EALDH1A1GLAHPGD
SCHEMBL21276083 0.68 POLB (0.43) ALDH1A1MAPK1
SCHEMBL24691517 0.68 MTHFD1 (0.46) ERN1DRD4DRD2DRD3
SCHEMBL20208889 0.67 MTHFD1 (0.47) ERN1DRD4DRD2DRD3
SCHEMBL17601909 0.67 ERN1 (1.00) ERN1DRD4DRD2DRD3
SCHEMBL6937223 0.66 SHBG (0.55) GAAKDM4EALDH1A1MAPK1SHBG
SCHEMBL31454878 0.65 ERN1 (0.79) GAAKDM4EALDH1A1GLAHPGD
SCHEMBL20209014 0.65 ERN1 (0.69) GAAKDM4EALDH1A1GLAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018097162-A1 SULFONAMIDE DERIVATIVE HAVING COUMARIN SKELETON 第一三共株式会社 2018-05-31 WO disclosed