SCHEMBL20208889

SCHEMBL20208889

Cc1c(OSC(F)(F)F)ccc2c3c(c(=O)oc12)CN(C(=O)OCc1ccccc1)CC3

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MTHFD1 P11586 2/20 0.47
MTHFD2 P13995 2/20 0.47
ERN1 O75460 5/20 0.46
PTGDR2 Q9Y5Y4 11/20 0.45
DRD2 P14416 1/20 0.44
DRD4 P21917 1/20 0.44
DRD3 P35462 1/20 0.44
FHIT P49789 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21354138 0.88 MTHFD1 (0.47) MTHFD1MTHFD2ERN1PTGDR2DRD2
SCHEMBL24691517 0.87 MTHFD1 (0.46) MTHFD1MTHFD2ERN1PTGDR2DRD2
SCHEMBL20208622 0.84 HSD17B10 (0.49) MTHFD1MTHFD2ERN1FHIT
SCHEMBL21354099 0.84 ERN1 (0.58) MTHFD1MTHFD2ERN1PTGDR2DRD2
SCHEMBL20208640 0.82 ERN1 (0.49) MTHFD1MTHFD2ERN1PTGDR2DRD2
SCHEMBL21417110 0.78 TMEM97 (0.49) MTHFD1MTHFD2ERN1
SCHEMBL20208684 0.74 CXCR3 (0.47) MTHFD1MTHFD2ERN1
SCHEMBL18928246 0.73 PTGDR2 (0.45) PTGDR2
SCHEMBL21354096 0.72 MTHFD2 (0.48) MTHFD1MTHFD2ERN1FHIT
SCHEMBL21354142 0.72 MTHFD2 (0.51) MTHFD1MTHFD2ERN1FHIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3546463-B1 SULFONAMIDE DERIVATIVE HAVING COUMARIN SKELETON DAIICHI SANKYO CO LTD (JP) 2022-12-07 EP disclosed
EP-3546463-A1 SULFONAMIDE DERIVATIVE HAVING COUMARIN SKELETON Daiichi Sankyo Co., Ltd. (JP) 2019-10-02 EP disclosed
WO-2018097162-A1 SULFONAMIDE DERIVATIVE HAVING COUMARIN SKELETON 第一三共株式会社 2018-05-31 WO disclosed