SCHEMBL20215217

SCHEMBL20215217

O=c1ccn(Cc2ccc(F)cc2)c(-c2cccc(C(F)(F)F)c2Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 7/20 0.43
MAPT P10636 2/20 0.40
THRB P10828 1/20 0.40
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NOTUM Q6P988 1/20 0.37
NR1H2 P55055 2/20 0.37
NR1H3 Q13133 2/20 0.37
ALDH1A1 P00352 2/20 0.36
CHRM5 P08912 2/20 0.36
CHRM3 P20309 1/20 0.36
ALDH2 P05091 1/20 0.35
ALDH3A1 P30838 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20215244 0.92 MAPT (0.39) P2RX7MAPTTHRBLMNANOTUM
SCHEMBL20215230 0.91 MAPK14 (0.43) P2RX7MAPTTHRBSMN1; SMN2NOTUM
SCHEMBL20215257 0.91 CHRM5 (0.46) P2RX7MAPTSMN1; SMN2NOTUMNR1H2
SCHEMBL20215219 0.91 P2RX7 (0.41) P2RX7MAPTLMNANOTUMALDH1A1
SCHEMBL20215232 0.90 MAPT (0.47) P2RX7MAPTTHRBLMNANOTUM
SCHEMBL20215246 0.89 PPARG (0.37) P2RX7NOTUMALDH1A1CHRM5
SCHEMBL20215256 0.87 KDM4E (0.43) P2RX7MAPTTHRBLMNASMN1; SMN2
SCHEMBL20215254 0.87 HCRTR1 (0.41) P2RX7MAPTNOTUMCHRM5CHRM3
SCHEMBL20215227 0.87 CYP11B1 (0.39) NOTUMALDH1A1
SCHEMBL20215242 0.87 MAPT (0.46) P2RX7MAPTLMNACHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9988373-B2 Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. (JP) 2018-06-05 US disclosed
US-9988373-B2 Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. (JP) 2018-06-05 US disclosed