SCHEMBL20215230

SCHEMBL20215230

O=c1ccn(Cc2cccc(F)c2)c(-c2cccc(C(F)(F)F)c2Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.43
POLB P06746 1/20 0.42
THRB P10828 1/20 0.42
EPHX2 P34913 4/20 0.41
DBH P09172 1/20 0.40
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
PKM P14618 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PPARG P37231 3/20 0.37
UBE2N P61088 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CA12 O43570 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
MAPT P10636 1/20 0.37
P2RX7 Q99572 3/20 0.36
AR P10275 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20215217 0.91 P2RX7 (0.43) THRBALDH1A1SMN1; SMN2MAPTP2RX7
SCHEMBL20215219 0.91 P2RX7 (0.41) MAPK14POLBALDH1A1MAPTP2RX7
SCHEMBL20215256 0.90 KDM4E (0.43) POLBTHRBDBHKDM4EMEN1
SCHEMBL20215253 0.89 MAPT (0.49) KDM4EALDH1A1KMT2ASMN1; SMN2CA12
SCHEMBL20215238 0.88 S1PR1 (0.36) POLBEPHX2KDM4EALDH1A1MAPT
SCHEMBL20215231 0.88 MAPT (0.46) POLBKDM4EMEN1ALDH1A1KMT2A
SCHEMBL20215244 0.87 MAPT (0.39) POLBTHRBKDM4EALDH1A1MAPT
SCHEMBL20215265 0.87 ALDH1A1 (0.40) MAPK14POLBALDH1A1MAPTP2RX7
SCHEMBL20215257 0.86 CHRM5 (0.46) KDM4EALDH1A1SMN1; SMN2CA12CA9
SCHEMBL20215232 0.85 MAPT (0.47) POLBTHRBKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9988373-B2 Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. (JP) 2018-06-05 US disclosed
US-9988373-B2 Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same SHIONOGI & CO., LTD. (JP) 2018-06-05 US disclosed