SCHEMBL20217424

SCHEMBL20217424

Cc1n[nH]c2ccc(NC(=O)C(c3ccccn3)C3CCCC3)cc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1E P28566 3/20 0.45
S1PR3 Q99500 3/20 0.45
FFAR2 O15552 1/20 0.45
MEN1 O00255 2/20 0.43
LMNA P02545 2/20 0.43
KMT2A Q03164 2/20 0.43
HTT P42858 2/20 0.43
PDPK1 O15530 3/20 0.43
ITK Q08881 3/20 0.42
CYP3A4 P08684 2/20 0.41
TTK P33981 2/20 0.41
AURKB Q96GD4 2/20 0.41
INCENP Q9NQS7 2/20 0.41
MAPT P10636 1/20 0.41
LRRK2 Q5S007 3/20 0.41
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ULK1 O75385 1/20 0.40
EGFR P00533 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14863447 0.88 FFAR2 (0.45) HTR1ES1PR3FFAR2MEN1LMNA
SCHEMBL14863461 0.84 FFAR2 (0.48) FFAR2PDPK1ITKCYP3A4TTK
SCHEMBL14863451 0.84 FFAR2 (0.48) FFAR2PDPK1ITKCYP3A4TTK
SCHEMBL14863553 0.84 FFAR2 (0.48) FFAR2PDPK1ITKCYP3A4TTK
SCHEMBL15477042 0.81 CYP3A4 (0.55) CYP3A4TTKAURKBINCENP
SCHEMBL15476924 0.78 TTK (0.67) PDPK1ITKCYP3A4TTKAURKB
SCHEMBL20217169 0.75 HTR1E (0.40) HTR1ES1PR3FFAR2MEN1LMNA
SCHEMBL20217418 0.74 FFAR2 (0.45) HTR1ES1PR3FFAR2MEN1LMNA
SCHEMBL14863558 0.72 ULK1 (0.45) HTR1ES1PR3MEN1LMNAKMT2A
SCHEMBL14863487 0.72 HTR1E (0.43) HTR1ES1PR3MEN1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2766352-B1 INDAZOLE COMPOUNDS AS KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIV HEALTH NETWORK UHN (CA) 2018-06-06 EP disclosed