SCHEMBL20217804

SCHEMBL20217804

N=C(c1ccc(N2C3CCC2CC(O)C3)cc1)c1cc(C(=O)NCc2ccccn2)ccc1N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.43
KDM4E B2RXH2 3/20 0.42
CYP3A4 P08684 2/20 0.42
TTK P33981 1/20 0.42
AURKB Q96GD4 1/20 0.42
INCENP Q9NQS7 1/20 0.42
NPC1 O15118 2/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
CYP1A2 P05177 1/20 0.41
CA2 P00918 1/20 0.41
NAMPT P43490 2/20 0.41
ALDH1A1 P00352 2/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 2/20 0.40
ROCK2 O75116 1/20 0.40
MEN1 O00255 1/20 0.40
MAPK14 Q16539 1/20 0.40
MELK Q14680 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20217341 0.91 CYP3A4 (0.40) RAB9ACYP3A4TTKAURKBINCENP
SCHEMBL20217630 0.90 RAB9A (0.45) RAB9AKDM4ECYP3A4TTKAURKB
SCHEMBL20217423 0.84 KDM4E (0.40) RAB9AKDM4ECYP3A4NPC1LMNA
SCHEMBL20217636 0.82 NAMPT (0.39) CA2NAMPTMAPK1ROCK2
SCHEMBL20217434 0.80 RAB9A (0.40) RAB9AKDM4ENPC1LMNAPOLB
SCHEMBL20217432 0.80 KMT2A (0.47) RAB9AKDM4ECYP3A4NPC1LMNA
SCHEMBL20217777 0.79 KMT2A (0.49) RAB9AKDM4ECYP3A4NPC1LMNA
SCHEMBL20217644 0.79 KMT2A (0.45) RAB9AKDM4ECYP3A4NPC1LMNA
SCHEMBL20217401 0.79 KDM4E (0.44) RAB9AKDM4ECYP3A4NPC1LMNA
SCHEMBL20217510 0.77 NAMPT (0.42) RAB9AKDM4ECYP3A4NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2766352-B1 INDAZOLE COMPOUNDS AS KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIV HEALTH NETWORK UHN (CA) 2018-06-06 EP disclosed