SCHEMBL20224587

SCHEMBL20224587

CCCc1ccc(-c2ccc(OS(=O)(=O)C(F)(F)F)c(F)c2F)cc1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MPL P40238 2/20 0.36
RARB P10826 1/20 0.35
DRD2 P14416 4/20 0.35
DRD3 P35462 4/20 0.35
DRD1 P21728 3/20 0.35
DRD4 P21917 3/20 0.35
DRD5 P21918 3/20 0.35
CA2 P00918 2/20 0.35
CA1 P00915 1/20 0.35
FFAR4 Q5NUL3 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRB2 P47870 1/20 0.34
HTR1D P28221 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13235229 0.89 MPL (0.34) MPLRARBDRD2DRD3DRD1
SCHEMBL20061708 0.81 RARB (0.43) RARBDRD2DRD3DRD1DRD4
SCHEMBL13198676 0.79 RARB (0.38) RARBDRD2DRD3DRD1DRD4
SCHEMBL20023230 0.79 CTSS (0.39) MPLRARBFFAR4GABRA1GABRB2
SCHEMBL29150477 0.78 DRD2 (0.36) DRD2DRD3DRD1DRD4DRD5
SCHEMBL2942703 0.78 MCL1 (0.41) RARBDRD2DRD3DRD1DRD4
SCHEMBL29873595 0.78 GABRA1 (0.42) MPLRARBFFAR4GABRA1GABRB2
SCHEMBL17616201 0.78 GABRA1 (0.46) MPLRARBFFAR4GABRA1GABRB2
SCHEMBL3437380 0.78 GABRA1 (0.42) MPLRARBFFAR4GABRA1GABRB2
SCHEMBL28328524 0.77 DGAT1 (0.38) MPLFFAR4GABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018100019-A1 THIOETHER-COMPOUNDS MERCK PATENT GMBH (DE) 2018-06-07 WO disclosed