SCHEMBL20253447

SCHEMBL20253447

Cc1cn(C)cc1S(N)(=O)=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 9/20 0.52
CA2 P00918 9/20 0.52
CA12 O43570 8/20 0.52
CA9 Q16790 8/20 0.52
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
GAA P10253 1/20 0.37
PDIA6 Q15084 1/20 0.34
CA6 P23280 3/20 0.33
CA5A P35218 2/20 0.33
CA7 P43166 2/20 0.33
CA5B Q9Y2D0 2/20 0.33
CA3 P07451 1/20 0.33
LMNA P02545 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CA4 P22748 2/20 0.32
CYP2C9 P11712 2/20 0.32
CA14 Q9ULX7 1/20 0.32
APEX1 P27695 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20253439 0.77 CA12 (0.34) CA1CA2CA12CA9
SCHEMBL348022 0.68
SCHEMBL6630171 0.67
SCHEMBL11511279 0.65 KDM4E (0.52) CA1CA2CA12CA9ALDH1A1
SCHEMBL4760209 0.65 KMT2A (0.47) CA1CA2CA12CA9ALDH1A1
SCHEMBL24696888 0.65 ALDH1A1 (0.41) CA1CA2CA12CA9ALDH1A1
SCHEMBL28827972 0.64 ALDH1A1 (0.50) CA1CA2CA12CA9ALDH1A1
SCHEMBL4544361 0.62
SCHEMBL23043571 0.62 ALDH1A1 (0.52) CA1CA2CA12CA9ALDH1A1
SCHEMBL7369 0.62 CA2 (0.56) CA1CA2CA12CA9PDIA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180162839-A1 Modulator of the Cystic Fibrosis Transmembrane Conductance Regulator, Pharmaceutical Compositions, Methods of Treatment, and Process for Making the Modulator VERTEX PHARMACEUTICALS (SAN DIEGO) LLC 2018-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180162839-A1 Modulator of the Cystic Fibrosis Transmembrane Conductance Regulator, Pharmaceutical Compositions, Methods of Treatment, and Process for Making the Modulator CFTR, SLC26A4, TMEM109 CA1 4518/4885CA2 1395/4885CA12 3191/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.