SCHEMBL20274172

SCHEMBL20274172

CC(c1cc2cc(F)ccc2o1)N1CCN(C(=O)CO)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.38
ALDH1A1 P00352 3/20 0.38
SIGMAR1 Q99720 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
CHRNA7 P36544 1/20 0.36
CACNA2D1 P54289 1/20 0.36
CACNA1B Q00975 1/20 0.36
CACNB1 Q02641 1/20 0.36
CACNA1C Q13936 1/20 0.36
F2 P00734 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20274131 0.86 HRH4 (0.48) ALDH1A1HRH3CYP2C9TSHRCACNA2D1
SCHEMBL20274215 0.85 PIM1 (0.43) POLBHRH3CACNA2D1CACNA1BCACNB1
SCHEMBL20274187 0.80 ALDH1A1 (0.45) POLBALDH1A1SIGMAR1HRH3CYP2D6
SCHEMBL15750162 0.78 F2 (0.57) ALDH1A1F2TPSAB1TPSD1TPSG1
SCHEMBL20274152 0.76 HTR2B (0.43) HRH3CYP2D6CYP2C9ALOX15TSHR
SCHEMBL15750158 0.70 PIM1 (0.41) POLBHRH3CACNA2D1CACNA1BCACNB1
SCHEMBL20274167 0.68 HRH3 (0.38) POLBHRH3CYP2D6CYP2C9ALOX15
SCHEMBL20274161 0.67 KCNH2 (0.52) CYP2D6CYP2C9ALOX15TSHRCYP2C19
SCHEMBL4792814 0.67 NPC1 (0.47) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL20274116 0.67 POLB (0.54) POLBALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3428162-B1 ANTHELMINTIC COMPOUNDS AND COMPOSITIONS AND METHOD OF USING THEREOF BOEHRINGER INGELHEIM ANIMAL HEALTH USA INC (US) 2021-05-05 EP disclosed
EP-2922845-B1 ANTHELMINTIC COMPOUNDS AND COMPOSITIONS AND METHOD OF USING THEREOF MERIAL INC (US) 2018-06-20 EP disclosed