SCHEMBL20277616

SCHEMBL20277616

NC(=O)C(Cc1ccccc1)NC(=O)c1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 6/20 0.71
CA1 P00915 2/20 0.62
CA12 O43570 1/20 0.62
CA9 Q16790 1/20 0.62
CTSL P07711 3/20 0.61
CTSS P25774 1/20 0.61
CTSK P43235 1/20 0.61
CA2 P00918 2/20 0.59
ACE P12821 2/20 0.59
PTPN1 P18031 1/20 0.58
CTRB1 P17538 3/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17244326 1.00 HPGDS (0.71) HPGDSCA1CA12CA9CTSL
SCHEMBL11425335 0.91 HPGDS (0.68) HPGDSCA1CA12CA9CTSL
SCHEMBL11781402 0.91 HPGDS (0.68) HPGDSCA1CA12CA9CTSL
SCHEMBL4684065 0.90 HPGDS (0.65) HPGDSCA1CA12CA9CTSL
SCHEMBL27002688 0.90 HPGDS (0.65) HPGDSCA1CA12CA9CTSL
SCHEMBL2105972 0.90 HPGDS (0.65) HPGDSCA1CA12CA9CTSL
SCHEMBL12320657 0.90 HPGDS (0.64) HPGDSCA1CA12CA9CA2
SCHEMBL27695921 0.90 HPGDS (0.65) HPGDSCA1CA12CA9CTSL
Hydrochloric Acid SCHEMBL7275137 0.88 HPGDS (0.67) HPGDSCA1CA12CA9CA2
SCHEMBL8443478 0.87 CTSL (0.62) HPGDSCA1CTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068405-B1 PYRROLO [1,2,F][1,2,4]TRIAZINES USEFUL FOR TREATING RESPIRATORY SYNCITIAL VIRUS INFECTIONS GILEAD SCIENCES INC (US) 2019-05-01 EP claimed
EP-4419513-B1 ANTITUMORAL COMPOUNDS PHARMA MAR SA (ES) 2025-08-27 EP disclosed
US-12384800-B2 Antitumoral compounds PHARMA MAR, S.A. (ES) 2025-08-12 US disclosed
US-20250243174-A1 ANTITUMORAL COMPOUNDS PHARMA MAR, S.A. (ES) 2025-07-31 US disclosed
EP-4419513-A1 ANTITUMORAL COMPOUNDS Pharma Mar S.A. (ES) 2024-08-28 EP disclosed
EP-4403042-A2 FLAVOR COMPOSITIONS AND PET FOOD PRODUCTS CONTAINING THE SAME Mars, Incorporated (US) 2024-07-24 EP disclosed
EP-3229612-B1 USE OF FLAVOR COMPOSITIONS AND PET FOOD PRODUCTS CONTAINING THE SAME MARS INC (US) 2024-06-26 EP disclosed
CN-118139851-A Antitumor compounds 法马马有限公司 2024-06-04 CN disclosed
US-20240166666-A1 ANTITUMORAL COMPOUNDS PHARMA MAR SA (ES) 2024-05-23 US disclosed
US-20240131180-A1 DRUG ANTIBODY CONJUGATES PHARMA MAR, S.A. (ES) 2024-04-25 US disclosed
US-10538535-B2 Antitumoral compounds PHARMA MAR, S.A. (ES) 2020-01-21 US disclosed
US-10442820-B2 2019-10-15 US disclosed
US-20190021380-A1 FLAVOR COMPOSITIONS AND PET FOOD PRODUCTS CONTAINING THE SAME MARS, INCORPORATED (US) 2019-01-24 US disclosed
US-20180312529-A1 Antitumoral Compounds PHARMA MAR, S.A. (ES) 2018-11-01 US disclosed
WO-2018197663-A1 ANTITUMORAL COMPOUNDS PHARMA MAR, S.A. (ES) 2018-11-01 WO disclosed
US-20180168208-A1 FLAVOR COMPOSITIONS AND PET FOOD PRODUCTS CONTAINING THE SAME MARS, INCORPORATED (US) 2018-06-21 US disclosed
US-20180168208-A1 FLAVOR COMPOSITIONS AND PET FOOD PRODUCTS CONTAINING THE SAME MARS, INCORPORATED (US) 2018-06-21 US disclosed
CN-102209532-B Method for reducing small, dense LDL particles METABOLEX INC 2015-07-22 CN disclosed
CN-101184726-B 2-arylpropionic acid derivatives and pharmaceutical compositions containing them DOMPE PHA R MA SPA RES & MFG 2012-05-30 CN disclosed
CN-101184726-A 2-arylpropionic acid derivatives and pharmaceutical compositions containing them DOMPE PHA R MA SPA RES & MFG (IT) 2008-05-21 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12384800-B2 Antitumoral compounds TP53, TOP1, MCL1 HPGDS 169/4885CA1 567/4885CA12 277/4885
US-10538535-B2 Antitumoral compounds TP53, RB1, XPOT HPGDS 2407/4885CA1 1866/4885CA12 1191/4885
US-20250243174-A1 ANTITUMORAL COMPOUNDS MCL1, XPOT, GZMB HPGDS 1144/4885CA1 945/4885CA12 305/4885
US-20240131180-A1 DRUG ANTIBODY CONJUGATES STT3B, STT3A, TTL HPGDS 942/4885CA1 2782/4885CA12 1331/4885
US-10442820-B2 RPS4X, RPS4Y1, XPOT HPGDS 2415/4885CA1 2834/4885CA12 1419/4885
US-20240166666-A1 ANTITUMORAL COMPOUNDS TP53, TOP1, MCL1 HPGDS 169/4885CA1 567/4885CA12 277/4885
US-20180312529-A1 Antitumoral Compounds TP53, RB1, XPOT HPGDS 2407/4885CA1 1866/4885CA12 1191/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.