SCHEMBL20288786

SCHEMBL20288786

CCCC(=O)NC(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.43
CA7 P43166 2/20 0.43
CA12 O43570 2/20 0.43
CA14 Q9ULX7 2/20 0.43
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
CTSD P07339 1/20 0.41
APLNR P35414 1/20 0.40
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
MAPT P10636 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CA2 P00918 2/20 0.38
CTSK P43235 6/20 0.38
CTSS P25774 3/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7557516 0.88 MAPT (0.44) CA1CA7CA12CA14APLNR
SCHEMBL7425805 0.86 HSP90AA1 (0.47) CA1CA7CA12CA14APLNR
SCHEMBL9424991 0.86 APLNR (0.39) CA1CA7CA12CA14APLNR
SCHEMBL240769 0.83 CA1 (0.42) CA1CA7CA12CA14APLNR
SCHEMBL17338702 0.82 APLNR (0.39) CA1CA7CA12CA14APLNR
SCHEMBL7052487 0.82 APLNR (0.54) CA1CA7CA12CA14HDAC3
SCHEMBL1261150 0.82 CYP2D6 (0.40) CA1CA7CA12CA14APLNR
SCHEMBL1262568 0.82 PHF8 (0.42) CA1CA7CA12CA14APLNR
SCHEMBL23461797 0.80 TDP1 (0.53) CA1CA7CA12CA14APLNR
SCHEMBL6463631 0.80 HDAC3 (0.40) CA1CA7CA12CA14HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018111805-A1 TETRAHYDROQUINOLINE-BASED BROMODOMAIN INHIBITORS ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2018-06-21 WO disclosed
CN-104080783-A Pyrrole compounds YAKULT HONSHA KK 2014-10-01 CN disclosed