SCHEMBL7557516

SCHEMBL7557516

CCCCC(=O)NC(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.44
ALDH1A1 P00352 4/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
KDM4E B2RXH2 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
PKM P14618 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CTSK P43235 5/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA7 P43166 1/20 0.41
CA14 Q9ULX7 1/20 0.41
APLNR P35414 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CTSS P25774 1/20 0.40
CAPN1 P07384 1/20 0.40
HSP90AA1 P07900 1/20 0.39
GAA P10253 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7425805 0.94 HSP90AA1 (0.47) MAPTALDH1A1KMT2AMEN1KDM4E
SCHEMBL20288786 0.88 CA1 (0.43) MAPTALDH1A1KMT2AMEN1NPSR1
SCHEMBL23461797 0.85 TDP1 (0.53) KMT2AMEN1CTSKCA12CA1
SCHEMBL5672978 0.83 TDP1 (0.40) KMT2AMEN1NPSR1CTSKCA12
SCHEMBL28755464 0.83 MAOA (0.45) ALDH1A1KMT2AMEN1CTSKCA1
SCHEMBL23461661 0.83 TDP1 (0.56) ALDH1A1KMT2AMEN1CTSKCA1
SCHEMBL13650887 0.83 TDP1 (0.40) ALDH1A1KMT2AMEN1PKMCTSK
SCHEMBL19485970 0.82 ZDHHC7 (0.42) KMT2AMEN1CTSKCTSSHSP90AA1
SCHEMBL14668808 0.81 CTSK (0.40) KMT2AMEN1CTSKCA12CA1
SCHEMBL5355236 0.81 GAA (0.47) ALDH1A1KMT2AMEN1CTSKGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111094233-B Compounds, compositions, and methods 戴纳立制药公司 2024-03-15 CN disclosed
EP-1171127-A2 PHARMACEUTICAL COMPOSITIONS CONTAINING PYRIDINE OR PYRIMIDINE DERIVATIVES FOR INHIBITION OF CYTOKINE PRODUCTION AND SECRETION Targacept, Inc. (US) 2002-01-16 EP disclosed
WO-2000062767-A2 PHARMACEUTICAL COMPOSITIONS CONTAINING PYRIDINE OR PYRIMIDINE DERIVATES FOR INHIBITION OF CYTOKINE PRODUCTION AND SECRETION TARGACEPT, INC. (US) 2000-10-26 WO disclosed