SCHEMBL20299487

SCHEMBL20299487

O=C1C(=Cc2ccc(C(F)(F)F)cc2)C(=O)c2ccccc21

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 2/20 0.51
CYP1A2 P05177 1/20 0.51
ITGA4 P13612 1/20 0.50
ITGB7 P26010 1/20 0.50
KMT2A Q03164 4/20 0.46
MAPT P10636 3/20 0.46
PIM1 P11309 1/20 0.46
PIM2 Q9P1W9 1/20 0.46
USP2 O75604 1/20 0.46
PKM P14618 1/20 0.46
ALDH1A1 P00352 3/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
NR1H3 Q13133 1/20 0.46
APP P05067 1/20 0.44
MAOB P27338 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
MEN1 O00255 1/20 0.44
ALPL P05186 1/20 0.44
ALPI P09923 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22625286 0.84 LCK (0.66) LCKKMT2AMAPTUSP2PKM
SCHEMBL28405872 0.82 ALDH1A1 (0.53) LCKKMT2AMAPTUSP2PKM
SCHEMBL30381597 0.79 PARP1 (0.62) LCKKMT2AMAPTUSP2PKM
SCHEMBL7147011 0.79 PARP1 (0.62) LCKKMT2AMAPTUSP2PKM
SCHEMBL677432 0.78 MAPT (0.62) LCKKMT2AMAPTUSP2PKM
SCHEMBL8483910 0.78 KDR (0.71) CYP1A2ITGA4ITGB7KMT2AMAPT
SCHEMBL8483914 0.78 KDR (0.71) CYP1A2ITGA4ITGB7KMT2AMAPT
SCHEMBL4157456 0.77 CYP19A1 (0.46) CYP1A2ITGA4ITGB7MAPTPIM1
SCHEMBL8072577 0.77 MAOA (0.49) LCKCYP1A2ITGA4ITGB7MAPT
SCHEMBL3372898 0.76 LCK (0.56) LCKKMT2AMAPTUSP2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110028407-B Method for preparing spiro [ cyclopropane-1, 2 ' -indene ] -1 ', 3 ' -diketone compound 苏州大学 2021-08-27 CN disclosed
WO-2020223439-A1 AURONES AND METHODS OF USING AURONES TO TREAT TUBERCULOSIS Middle Tennessee State University (US) 2020-11-05 WO disclosed
WO-2018114965-A1 CLPX INHIBITORY COMPOUNDS FOR THE TREATMENT OF MULTI RESISTANT STAPHYLOCOCCUS AUREUS VIRULENCE AND FOR THE TREATMENT OF LEUKEMIA Technische Universität München (DE) 2018-06-28 WO disclosed