SCHEMBL2033213

SCHEMBL2033213

O=C1C=C(Nc2ccccc2)CCC1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MT-CO2 P00403 1/20 0.69
MEN1 O00255 1/20 0.58
KMT2A Q03164 1/20 0.58
POLB P06746 2/20 0.57
SMN1; SMN2 Q16637 3/20 0.51
MAPK1 P28482 2/20 0.51
GAA P10253 1/20 0.44
LMNA P02545 2/20 0.43
MAPT P10636 2/20 0.43
ATM Q13315 1/20 0.43
ALDH1A1 P00352 3/20 0.42
TDP1 Q9NUW8 2/20 0.42
RAB9A P51151 1/20 0.41
HSD17B10 Q99714 2/20 0.41
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
ALOX12 P18054 1/20 0.39
PTGS1 P23219 1/20 0.39
SLC6A2 P23975 1/20 0.39
PTGS2 P35354 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10811051 0.88 MT-CO2 (0.58) MT-CO2MEN1KMT2APOLBSMN1; SMN2
SCHEMBL6583074 0.83 POLB (0.56) MT-CO2MEN1KMT2APOLBSMN1; SMN2
SCHEMBL9275585 0.81 MT-CO2 (0.70) MT-CO2MEN1KMT2APOLBSMN1; SMN2
SCHEMBL9596455 0.80 MT-CO2 (0.54) MT-CO2MEN1KMT2APOLBSMN1; SMN2
SCHEMBL15102230 0.80 IDH2 (0.50) MT-CO2MEN1KMT2APOLBMAPK1
SCHEMBL16784518 0.79 MEN1 (0.73) MT-CO2MEN1KMT2APOLBSMN1; SMN2
SCHEMBL16391829 0.79 ABCG2 (0.51) MT-CO2MEN1KMT2APOLBRAB9A
SCHEMBL3988142 0.77 KMT2A (0.65) MT-CO2MEN1KMT2APOLBMAPK1
SCHEMBL15992015 0.76 MT-CO2 (0.50) MT-CO2MEN1KMT2APOLBSMN1; SMN2
SCHEMBL15992074 0.76 KIF11 (0.52) MT-CO2SMN1; SMN2GAAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110713454-A Nitro-substituted indole compound and preparation method thereof 南京工业大学 2020-01-21 CN claimed
EP-0214009-A2 Enaminones as potential prodrugs of primary and secondary amines MERCK & CO. INC. (US) 1987-03-11 EP claimed
CN-110713454-A Nitro-substituted indole compound and preparation method thereof 南京工业大学 2020-01-21 CN disclosed
EP-2509954-A1 4 -OXO- 1H -QUINOLINE- 3 - CARBOXAMIDES AS MODULATORS OF ATP -BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2012-10-17 EP disclosed
WO-2011072241-A1 4 -OXO- IH -QUINOLINE- 3 - CARBOXAMIDES AS MODULATORS OF ATP -BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-06-16 WO disclosed
EP-0214009-A2 Enaminones as potential prodrugs of primary and secondary amines MERCK & CO. INC. (US) 1987-03-11 EP disclosed