SCHEMBL20344808

SCHEMBL20344808

CCc1c(C)cn2cc(-c3cccc(-c4ccccc4F)c3)nc2c1-c1ccc2c(c1)CCCO2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GNRHR P30968 1/20 0.35
FABP4 P15090 6/20 0.34
CTNNB1 P35222 2/20 0.33
WNT3A P56704 2/20 0.33
APP P05067 1/20 0.33
BACE1 P56817 1/20 0.33
KDM4E B2RXH2 3/20 0.32
RAB9A P51151 3/20 0.32
NPC1 O15118 2/20 0.32
MAPT P10636 2/20 0.32
PKM P14618 2/20 0.32
ALDH1A1 P00352 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
RIPK1 Q13546 1/20 0.32
AXL P30530 1/20 0.32
MERTK Q12866 1/20 0.32
STIM1 Q13586 1/20 0.31
ORAI1 Q96D31 1/20 0.31
PFKFB3 Q16875 1/20 0.31
WDR5 P61964 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20344816 0.91 APP (0.33) GNRHRFABP4APPBACE1KDM4E
SCHEMBL17039278 0.90 FABP4 (0.41) GNRHRFABP4CTNNB1WNT3ASMN1; SMN2
SCHEMBL17029029 0.81 NR1I2 (0.44) FABP4
SCHEMBL17039243 0.81 NR1I2 (0.44) FABP4
SCHEMBL17029048 0.81 NR1I2 (0.44) FABP4
SCHEMBL17039306 0.80 FABP4 (0.35) GNRHRFABP4RAB9ANPC1MAPT
SCHEMBL18364984 0.79 NR1I2 (0.39) FABP4FABP3
SCHEMBL17039253 0.79 NR1I2 (0.39) FABP4FABP3
SCHEMBL20344807 0.77 P2RX7 (0.33)
SCHEMBL17039255 0.75 CLK1 (0.40) FABP4KDM4ERAB9ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3107913-B1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV HEALTHCARE UK NO 5 LTD (GB) 2018-07-04 EP disclosed