SCHEMBL17039306

SCHEMBL17039306

COC(=O)Cc1c(C)cn2cc(-c3cccc(-c4ccc(F)c(F)c4F)c3)nc2c1-c1ccc2c(c1)CCCO2

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FABP4 P15090 5/20 0.35
FABP3 P05413 2/20 0.35
NPC1 O15118 1/20 0.34
CLK1 P49759 1/20 0.34
RAB9A P51151 1/20 0.34
EED O75530 3/20 0.33
RBBP4 Q09028 3/20 0.33
SUZ12 Q15022 3/20 0.33
EZH2 Q15910 3/20 0.33
AEBP2 Q6ZN18 3/20 0.33
MAPT P10636 1/20 0.33
P2RX7 Q99572 2/20 0.32
GNRHR P30968 1/20 0.32
KLKB1 P03952 2/20 0.32
GRM5 P41594 1/20 0.32
BRD4 O60885 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20344816 0.89 APP (0.33) FABP4FABP3NPC1CLK1RAB9A
SCHEMBL17039278 0.84 FABP4 (0.41) FABP4FABP3GNRHRGRM5
SCHEMBL20344817 0.83 NR1I2 (0.36) FABP4FABP3
SCHEMBL18364988 0.83 NR1I2 (0.36) FABP4FABP3
SCHEMBL17029028 0.82 NR1I2 (0.42) FABP4
SCHEMBL17029056 0.82 NR1I2 (0.42) FABP4
SCHEMBL17039255 0.81 CLK1 (0.40) FABP4FABP3NPC1CLK1RAB9A
SCHEMBL20344807 0.81 P2RX7 (0.33) P2RX7
SCHEMBL20344808 0.80 GNRHR (0.35) FABP4FABP3NPC1RAB9AMAPT
SCHEMBL20344786 0.78 P2RX7 (0.33) MAPTP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015126765-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BRISTOL-MYERS SQUIBB COMPANY (US) 2015-08-27 WO disclosed