SCHEMBL20346374

SCHEMBL20346374

CCOC(=O)Cc1ccc(C(=O)n2c(C)c(CC(=O)OCC)c3cc(C)ccc32)cc1

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.64
AKR1C3 P42330 6/20 0.60
AKR1C2 P52895 4/20 0.60
HTR1A P08908 1/20 0.53
PKM P14618 1/20 0.53
PTGS1 P23219 1/20 0.53
GLO1 Q04760 1/20 0.53
HIF1A Q16665 1/20 0.53
CNR2 P34972 1/20 0.53
AKR1C4 P17516 1/20 0.52
AKR1C1 Q04828 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20346373 0.90 PTGS2 (0.79) PTGS2AKR1C3HTR1APKMPTGS1
SCHEMBL20349624 0.88 PTGS2 (0.83) PTGS2AKR1C3AKR1C2HTR1APKM
SCHEMBL20346375 0.84 PTGS2 (0.62) PTGS2AKR1C3AKR1C2HTR1APKM
SCHEMBL13448804 0.83 AKR1C3 (0.83) PTGS2AKR1C3AKR1C2HIF1ACNR2
SCHEMBL17369628 0.80 PTGS2 (0.67) PTGS2AKR1C3AKR1C2HTR1APKM
SCHEMBL25873193 0.80 PTGS2 (0.80) PTGS2AKR1C3AKR1C2HTR1APKM
SCHEMBL17946351 0.79 AKR1C3 (0.78) PTGS2AKR1C3AKR1C2PTGS1GLO1
SCHEMBL4549122 0.78 PTGS2 (1.00) PTGS2AKR1C3AKR1C2HTR1APKM
SCHEMBL24890591 0.78 AKR1C3 (0.64) PTGS2AKR1C3AKR1C2CNR2
SCHEMBL16557623 0.78 AKR1C3 (0.71) PTGS2AKR1C3AKR1C2PTGS1GLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180186721-A1 OXIDATIVE COUPLING OF ARYL BORON REAGENTS WITH SP3-CARBON NUCLEOPHILES, AND AMBIENT DECARBOXYLATIVE ARYLATION OF MALONATE HALF-ESTERS VIA OXIDATIVE CATALYSIS THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2018-07-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180186721-A1 OXIDATIVE COUPLING OF ARYL BORON REAGENTS WITH SP3-CARBON NUCLEOPHILES, AND AMBIENT DECARBOXYLATIVE ARYLATION OF MALONATE HALF-ESTERS VIA OXIDATIVE CATALYSIS SOD1, AOC3, CBR3 PTGS2 3910/4885AKR1C3 47/4885AKR1C2 81/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.