SCHEMBL13448804

SCHEMBL13448804

COC(=O)Cc1c(C)n(C(=O)c2ccc(C)cc2)c2ccc(C)cc12

nearest known ligand 0.83

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 6/20 0.83
AKR1C2 P52895 3/20 0.83
PTGS2 P35354 11/20 0.69
CNR2 P34972 1/20 0.69
MAPT P10636 1/20 0.58
LMNA P02545 2/20 0.56
ALDH1A1 P00352 1/20 0.56
HPGD P15428 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
CYP1A2 P05177 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
TSHR P16473 1/20 0.55
NFKB1 P19838 1/20 0.55
HIF1A Q16665 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25873193 0.93 PTGS2 (0.80) AKR1C3AKR1C2PTGS2CNR2MAPT
SCHEMBL27768669 0.92 AKR1C3 (0.78) AKR1C3AKR1C2PTGS2CNR2MAPT
SCHEMBL16656482 0.91 AKR1C3 (1.00) AKR1C3AKR1C2PTGS2CNR2MAPT
SCHEMBL17946351 0.86 AKR1C3 (0.78) AKR1C3AKR1C2PTGS2MAPTLMNA
SCHEMBL20346374 0.83 PTGS2 (0.64) AKR1C3AKR1C2PTGS2CNR2HIF1A
SCHEMBL14983579 0.82 AKR1C3 (0.60) AKR1C3AKR1C2PTGS2MAPTLMNA
SCHEMBL20346373 0.82 PTGS2 (0.79) AKR1C3PTGS2CNR2HIF1A
SCHEMBL20259423 0.82 PTGS2 (0.78) AKR1C3AKR1C2PTGS2CNR2MAPT
SCHEMBL24890591 0.82 AKR1C3 (0.64) AKR1C3AKR1C2PTGS2CNR2MAPT
SCHEMBL30761037 0.82 AKR1C3 (0.87) AKR1C3AKR1C2PTGS2CNR2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9012647-B2 Nitroxide modified non-steroidal anti-inflammatory compounds and uses thereof in the treatment and prevention of diseases or disorders THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2015-04-21 US disclosed
US-20120263650-A1 NITROXIDE MODIFIED NON-STEROIDAL ANTI-INFLAMMATORY COMPOUNDS AND USES THEREOF IN THE TREATMENT AND PREVENTION OF DISEASES OR DISORDERS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH 2012-10-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120263650-A1 NITROXIDE MODIFIED NON-STEROIDAL ANTI-INFLAMMATORY COMPOUNDS AND USES THEREOF IN THE TREATMENT AND PREVENTION OF DISEASES OR DISORDERS NOS1, NOS3, PTGS1 AKR1C3 315/4885AKR1C2 415/4885PTGS2 12/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.