SCHEMBL20354517

SCHEMBL20354517

Cc1ccc2c(c1)CN(C)CCO2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.51
CREBBP Q92793 1/20 0.44
PIK3CA P42336 3/20 0.41
PIK3CB P42338 3/20 0.41
PIK3CG P48736 3/20 0.41
ALDH1A1 P00352 3/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
HSD17B10 Q99714 1/20 0.41
HTT P42858 1/20 0.41
DRD2 P14416 2/20 0.40
DRD1 P21728 2/20 0.40
DRD4 P21917 2/20 0.40
DRD5 P21918 2/20 0.40
DRD3 P35462 2/20 0.40
PKM P14618 3/20 0.40
KMT2A Q03164 2/20 0.40
HPGD P15428 2/20 0.40
POLB P06746 1/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20354516 0.86 DRD2 (0.47) RIPK1CREBBPPIK3CAPIK3CBPIK3CG
SCHEMBL24258522 0.84 CREBBP (0.65) RIPK1CREBBPPIK3CAPIK3CBPIK3CG
SCHEMBL676648 0.82 MAPT (0.42) RIPK1CREBBPALDH1A1GAAMAPT
SCHEMBL1950203 0.81 KDM4E (0.42) ALDH1A1GAAMAPTHTTDRD2
SCHEMBL14863559 0.81 HTT (0.43) RIPK1PIK3CAPIK3CBPIK3CGMAPT
Hydrochloric Acid SCHEMBL7481044 0.80 KDM4E (0.45) GAAMAPTHTTDRD2DRD1
SCHEMBL18255843 0.78 PIK3CA (0.43) RIPK1PIK3CAPIK3CBPIK3CGHTT
SCHEMBL5022145 0.77 KMT2A (0.52) CREBBPPIK3CAPIK3CBPIK3CGALDH1A1
SCHEMBL29388834 0.77 MAOA (0.53) HTTDRD2DRD1DRD4DRD5
SCHEMBL10455557 0.77 MAOA (0.53) HTTDRD2DRD1DRD4DRD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021028645-A1 PLASMA KALLIKREIN INHIBITORS KALVISTA PHARMACEUTICALS LIMITED (GB) 2021-02-18 WO disclosed
WO-2021028649-A1 PLASMA KALLIKREIN INHIBITORS KALVISTA PHARMACEUTICALS LIMITED (GB) 2021-02-18 WO disclosed
EP-3564232-A1 BMP-SIGNAL-INHIBITING COMPOUND Riken (JP) 2019-11-06 EP disclosed
WO-2018124001-A1 BMP-SIGNAL-INHIBITING COMPOUND 国立研究開発法人理化学研究所 2018-07-05 WO disclosed