SCHEMBL24258522

SCHEMBL24258522

Cc1ccc(C)c(-c2ccc3c(c2)CN(C)CCO3)c1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 14/20 0.65
APP P05067 1/20 0.44
BACE1 P56817 1/20 0.44
RIPK1 Q13546 1/20 0.40
PIK3CA P42336 4/20 0.40
PIK3CB P42338 3/20 0.40
PIK3CG P48736 3/20 0.40
PIK3CD O00329 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20354517 0.84 RIPK1 (0.51) CREBBPRIPK1PIK3CAPIK3CBPIK3CG
SCHEMBL19657514 0.79 CREBBP (1.00) CREBBP
SCHEMBL20354516 0.75 DRD2 (0.47) CREBBPRIPK1PIK3CAPIK3CBPIK3CG
SCHEMBL1950203 0.71 KDM4E (0.42)
SCHEMBL14863559 0.71 HTT (0.43) RIPK1PIK3CAPIK3CBPIK3CGPIK3CD
SCHEMBL23251650 0.70 PIK3CA (0.58) CREBBPPIK3CA
Hydrochloric Acid SCHEMBL7481044 0.70 KDM4E (0.45)
SCHEMBL14003406 0.69 KDM4E (0.54) CREBBPAPPBACE1
SCHEMBL676648 0.69 MAPT (0.42) CREBBPRIPK1
SCHEMBL18255843 0.68 PIK3CA (0.43) RIPK1PIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3464270-B1 HETEROCYCLIC INHIBITORS OF CBP/EP300 AND THEIR USE IN THE TREATMENT OF CANCER GENENTECH INC (US) 2022-02-23 EP disclosed