SCHEMBL2038048

SCHEMBL2038048

Cc1cc(OCC(F)(F)F)ccc1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.47
CYP2C9 P11712 2/20 0.45
CYP17A1 P05093 1/20 0.45
CYP2C19 P33261 1/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 2/20 0.43
MAPT P10636 3/20 0.43
GPR3 P46089 1/20 0.43
LMNA P02545 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
STAT3 P40763 1/20 0.43
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29972693 1.00 SMN1; SMN2 (0.47) SMN1; SMN2CYP2C9CYP17A1CYP2C19KDM4E
SCHEMBL17717291 0.83 SMN1; SMN2 (0.46) SMN1; SMN2CYP2C9CYP17A1CYP2C19MAPT
SCHEMBL24683493 0.83 CYP2C9 (0.49) SMN1; SMN2CYP2C9CYP17A1CYP2C19KDM4E
SCHEMBL12578461 0.81 SMN1; SMN2 (0.49) SMN1; SMN2MAPTLMNAALOX15TSHR
SCHEMBL29972592 0.80 KDM4E (0.45) SMN1; SMN2CYP2C9CYP17A1CYP2C19KDM4E
SCHEMBL23977879 0.80 CYP2C9 (0.46) SMN1; SMN2CYP2C9CYP17A1CYP2C19KDM4E
SCHEMBL14937673 0.80 KDM4E (0.45) SMN1; SMN2CYP2C9CYP17A1CYP2C19KDM4E
SCHEMBL23414843 0.80 KDM4E (0.45) SMN1; SMN2CYP2C9CYP17A1CYP2C19KDM4E
SCHEMBL2031055 0.80 ALDH1A1 (0.55) SMN1; SMN2CYP2C9CYP17A1CYP2C19KDM4E
SCHEMBL25405284 0.79 SMN1; SMN2 (0.53) SMN1; SMN2ALDH1A1MAPTLMNAALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12479844-B2 Ion channel modulators PRAXIS PRECISION MEDICINES, INC. (US) 2025-11-25 US disclosed
US-12473289-B2 Heterocyclic compounds as delta-5 desaturase inhibitors and methods of use AMGEN INC. (US) 2025-11-18 US disclosed
US-20250145637-A1 SULFONAMIDE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF JIANGSU HENGRUI PHARMACEUTICALS CO., LTD. (CN) 2025-05-08 US disclosed
EP-4385989-A1 SULFONAMIDE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF Jiangsu Hengrui Pharmaceuticals Co., Ltd. (CN) 2024-06-19 EP disclosed
CN-117597341-A Sulfonamide derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2024-02-23 CN disclosed
WO-2023016484-A1 SULFONAMIDE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 江苏恒瑞医药股份有限公司 2023-02-16 WO disclosed
WO-2023016484-A1 SULFONAMIDE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 江苏恒瑞医药股份有限公司 2023-02-16 WO disclosed
EP-4065579-A1 HETEROCYCLIC COMPOUNDS AS DELTA-5 DESATURASE INHIBITORS AND METHODS OF USE Amgen Inc. (US) 2022-10-05 EP disclosed
US-20210403476-A1 ION CHANNEL MODULATORS PRAXIS PRECISION MEDICINES, INC. 2021-12-30 US disclosed
CN-113573713-A Ion channel modulators 普拉克西斯精密药物股份有限公司 2021-10-29 CN disclosed
WO-2021108404-A1 HETEROCYCLIC COMPOUNDS AS DELTA-5 DESATURASE INHIBITORS AND METHODS OF USE AMGEN INC. (US) 2021-06-03 WO disclosed
WO-2020069322-A1 ION CHANNEL MODULATORS PRAXIS PRECISION MEDICINES, INC. (US) 2020-04-02 WO disclosed
EP-2079674-B1 PROCESS FOR THE PREPARATION OF TRIFLUOROETHOXYTOLUENES GRINDEKS JSC (LV) 2011-06-29 EP disclosed
US-20100063292-A1 PROCESS FOR THE PREPARATION OF TRIFLUOROETHOXYTOLUENES. GRINDEKS A JOINT STOCK COMPANY (LV) 2010-03-11 US disclosed
US-20100056794-A1 PROCESS FOR THE PREPARATION OF 2,5-BIS-(2,2,2-TRIFLUOROETHOXY)-N-(2-PIPERIDYL-METHYL)-BENZAMIDE AND SALTS THEREOF GRINDEKS A JOINT STOCK COMPANY (LV) 2010-03-04 US disclosed
EP-2079674-A1 PROCESS FOR THE PREPARATION OF TRIFLUOROETHOXYTOLUENES Grindeks, a joint stock company (LV) 2009-07-22 EP disclosed
EP-2079692-A1 PROCESS FOR THE PREPARATION OF 2,5-BIS-(2,2,2-TRIFLUOROETHOXY)-N-(2-PIPERIDYLMETHYL)-BENZAMIDE AND SALTS THEREOF Grindeks, a joint stock company (LV) 2009-07-22 EP disclosed
WO-2008055849-A1 PROCESS FOR THE PREPARATION OF TRIFLUOROETHOXYTOLUENES GRINDEKS, A JOINT STOCK COMPANY (LV) 2008-05-15 WO disclosed
WO-2008055851-A1 PROCESS FOR THE PREPARATION OF 2,5-BIS-(2,2,2-TRIFLUOROETHOXY)-N-(2-PIPERIDYLMETHYL)-BENZAMIDE AND SALTS THEREOF GRINDEKS, A JOINT STOCK COMPANY (LV) 2008-05-15 WO disclosed
EP-1918280-A1 Process for the preparation of 2,5-bis-(2,2,2-trifluoroethoxy)-N-(2-piperidylmethyl)-benzamide and salts thereof "Joint Stock Company Grindeks" (LV) 2008-05-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210403476-A1 ION CHANNEL MODULATORS SCN1A, SCN3A, SCN2A SMN1; SMN2 185/4885CYP2C9 3258/4885CYP17A1 4316/4885
US-20100056794-A1 PROCESS FOR THE PREPARATION OF 2,5-BIS-(2,2,2-TRIFLUOROETHOXY)-N-(2-PIPERIDYL-METHYL)-BENZAMIDE AND SALTS THEREOF BOLA2; BOLA2B, TET2, CYP1A2 SMN1; SMN2 1097/4885CYP2C9 181/4885CYP17A1 1481/4885
US-20250145637-A1 SULFONAMIDE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF SULT2A1, KAT8, TST SMN1; SMN2 4679/4885CYP2C9 648/4885CYP17A1 408/4885
US-12479844-B2 Ion channel modulators SCN1A, SCN3A, SCN2A SMN1; SMN2 185/4885CYP2C9 3258/4885CYP17A1 4316/4885
US-12473289-B2 Heterocyclic compounds as delta-5 desaturase inhibitors and methods of use SCD5, SCD, FADS2 SMN1; SMN2 3098/4885CYP2C9 116/4885CYP17A1 320/4885
US-20100063292-A1 PROCESS FOR THE PREPARATION OF TRIFLUOROETHOXYTOLUENES. CYP2C9, CYP3A4, CYP3A5 SMN1; SMN2 1342/4885CYP2C9 1/4885CYP17A1 1900/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.