SCHEMBL23912253

SCHEMBL23912253

CCc1nc2cccc(CCC=O)c2c(=O)n1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.45
ALDH1A1 P00352 1/20 0.45
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
USP2 O75604 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
PIK3CD O00329 2/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 1/20 0.41
PIK3R1 P27986 1/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20404284 0.83 SMN1; SMN2 (0.48) SMN1; SMN2ALDH1A1ESR1ESR2USP2
SCHEMBL23912254 0.82 PIK3CD (0.55) SMN1; SMN2ALDH1A1ESR1ESR2PIK3CD
SCHEMBL20404285 0.81 HDAC1 (0.50) SMN1; SMN2ALDH1A1ESR1ESR2USP2
SCHEMBL20404396 0.80 PIK3CD (0.57) SMN1; SMN2ALDH1A1ESR1ESR2USP2
SCHEMBL23912237 0.79 HRH3 (0.59) PIK3CDKCNH2HRH3
SCHEMBL17458010 0.79 PIK3CD (0.53) PIK3CDPIK3R1HDAC6
SCHEMBL16597182 0.78 SMN1; SMN2 (0.50) SMN1; SMN2ALDH1A1ESR1ESR2NPC1
SCHEMBL16597185 0.78 PDE10A (0.52) SMN1; SMN2ALDH1A1ESR1ESR2NPC1
SCHEMBL17235505 0.78 ESR1 (0.60) SMN1; SMN2ALDH1A1ESR1ESR2USP2
SCHEMBL23912240 0.78 PIK3CD (0.55) SMN1; SMN2ALDH1A1PIK3CDLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3160960-B1 PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS GILEAD SCIENCES INC (US) 2021-10-13 EP disclosed