SCHEMBL20405679

SCHEMBL20405679

C=C(/N=C(\OC)c1nnn(-c2ccccc2F)c1CCCC)c1ccccc1F

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 8/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
NPSR1 Q6W5P4 2/20 0.31
NR1I2 O75469 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ALDH1A1 P00352 2/20 0.31
LMNA P02545 2/20 0.31
USP2 O75604 1/20 0.31
TSHR P16473 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20405705 0.90 NPSR1 (0.35) KCNN4MEN1KMT2ANPSR1NR1I2
SCHEMBL13765502 0.81 KCNN4 (0.33) KCNN4MEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL2220115 0.75 HTT (0.42) KCNN4MEN1KMT2ANPSR1SMN1; SMN2
SCHEMBL20405685 0.75 HPGD (0.37) KCNN4MEN1KMT2ANPSR1SMN1; SMN2
SCHEMBL2219573 0.68 HTT (0.43) KCNN4MEN1KMT2ANPSR1SMN1; SMN2
SCHEMBL1423244 0.68 REN (0.40) KCNN4MEN1KMT2ANPSR1SMN1; SMN2
SCHEMBL13765447 0.66 DHODH (0.31) MEN1KMT2A
SCHEMBL13765531 0.66 IDH1 (0.35) NPSR1SMN1; SMN2ALDH1A1LMNATSHR
SCHEMBL3456050 0.66 KCNN4 (0.42) KCNN4NPSR1SMN1; SMN2ALDH1A1
SCHEMBL13765396 0.66 DRD2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250165-B1 TRIAZOLE OXADIAZOLES DERIVATIVES MERCK SERONO SA (CH) 2018-07-25 EP disclosed