Nitenpyram

Nitenpyram

SCHEMBL20425327

CCCC[SnH](CCCC)CCCC.CCN(Cc1ccc(Cl)nc1)/C(=C/[N+](=O)[O-])NC

nearest known ligand 0.83

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
MAPT P10636 2/20 0.36
FAAH O00519 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
CHRNA1 P02708 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA7 P36544 1/20 0.33
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
CASP6 P55212 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nitenpyram SCHEMBL25789 0.91 SMN1; SMN2 (0.40) ALDH1A1MAPTFAAHCYP3A4CYP2D6
Nitenpyram SCHEMBL13448342 0.91 SMN1; SMN2 (0.40) ALDH1A1MAPTFAAHCYP3A4CYP2D6
Nitenpyram SCHEMBL29388004 0.91 SMN1; SMN2 (0.40) ALDH1A1MAPTFAAHCYP3A4CYP2D6
Nitenpyram SCHEMBL31030931 0.91 SMN1; SMN2 (0.40) ALDH1A1MAPTFAAHCYP3A4CYP2D6
Nitenpyram SCHEMBL25788 0.91 SMN1; SMN2 (0.40) ALDH1A1MAPTFAAHCYP3A4CYP2D6
Nitenpyram SCHEMBL28400760 0.89 SMN1; SMN2 (0.39) ALDH1A1MAPTFAAHCYP3A4CYP2D6
SCHEMBL7660190 0.85 CHRNB2 (0.36) ALDH1A1MAPTFAAHCYP3A4CYP2D6
SCHEMBL7753555 0.85 CHRNB2 (0.36) ALDH1A1MAPTFAAHCYP3A4CYP2D6
SCHEMBL7668848 0.82 CHRNB2 (0.38) ALDH1A1MAPTCYP3A4CYP2D6CYP2C9
SCHEMBL7678862 0.81 ALDH1A1 (0.39) ALDH1A1MAPTFAAHCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3573638-A1 COMPOSITIONS AND RELATED METHODS FOR CONTROLLING VECTOR-BORNE DISEASES Flagship Pioneering Innovations V, Inc. (US) 2019-12-04 EP disclosed
EP-3573465-A1 METHODS AND RELATED COMPOSITIONS FOR MANUFACTURING FOOD AND FEED Flagship Pioneering Innovations V, Inc. (US) 2019-12-04 EP disclosed
WO-2018156998-A1 COMPOSITIONS AND RELATED METHODS FOR MODULATING ENDOSYMBIONTS FLAGSHIP PIONEERING, INC. (US) 2018-08-30 WO disclosed
WO-2018140496-A1 METHODS AND RELATED COMPOSITIONS FOR MANUFACTURING FOOD AND FEED FLAGSHIP PIONEERING, INC. (US) 2018-08-02 WO disclosed
WO-2018140479-A1 COMPOSITIONS AND RELATED METHODS FOR AGRICULTURE FLAGSHIP PIONEERING, INC. (US) 2018-08-02 WO disclosed
WO-2018140519-A1 COMPOSITIONS AND RELATED METHODS FOR AGRICULTURE FLAGSHIP PIONEERING, INC. (US) 2018-08-02 WO disclosed
WO-2018140507-A1 COMPOSITIONS AND RELATED METHODS FOR CONTROLLING VECTOR-BORNE DISEASES FLAGSHIP PIONEERING, INC. (US) 2018-08-02 WO disclosed